SCHEMBL22877153

SCHEMBL22877153

COc1cccc(OC)c1C1CCCC1N

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.50
ABCB1 P08183 1/20 0.42
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 1/20 0.41
HSD11B1 P28845 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37
HTR1A P08908 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6745026 0.81 HTR2C (0.51) HTR2AHTR2CHTR2BHSD11B1MEN1
SCHEMBL17356793 0.80 ABCB1 (0.43) ADRA1AABCB1DRD2HSD11B1CA1
SCHEMBL1643779 0.77 HTR2C (0.51) HTR2AHTR2CHTR2BHSD11B1MEN1
SCHEMBL1643778 0.77 HTR2C (0.51) HTR2AHTR2CHTR2BHSD11B1MEN1
SCHEMBL8439755 0.74 HTR2A (0.47) HTR2AHTR2CHTR2BHSD11B1
SCHEMBL17356807 0.72 HTR1A (0.40) ADRA1AABCB1DRD2HSD11B1CA1
SCHEMBL17356810 0.72 ADRA1A (0.42) ADRA1AABCB1DRD2CA1CA2
SCHEMBL6273883 0.71 ADRA1A (0.58) ADRA1AHTR2AHTR2CHTR2BKDM1A
SCHEMBL10263051 0.71 HTR2C (0.55) DRD2HTR2AHTR2CHTR2BKDM1A
SCHEMBL4259949 0.71 HTR2C (0.55) DRD2HTR2AHTR2CHTR2BKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107898-B1 1,2-SUBSTITUTED CYCLOPENTANES AS OREXIN RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICALS CO (JP) 2021-01-06 EP disclosed