SCHEMBL22883

SCHEMBL22883

Cc1nc2nc(N)[nH]c(=O)c2[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PNP P00491 5/20 0.73
KDM4E B2RXH2 1/20 0.58
MEN1 O00255 1/20 0.58
ALDH1A1 P00352 1/20 0.58
MAPT P10636 1/20 0.58
THRB P10828 1/20 0.58
HPGD P15428 1/20 0.58
KMT2A Q03164 1/20 0.58
HSD17B10 Q99714 1/20 0.58
FGFR1 P11362 3/20 0.51
FGFR2 P21802 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26155923 0.92 PNP (0.73) PNPKDM4EMEN1ALDH1A1MAPT
Trifluoroacetic Acid SCHEMBL2300171 0.86 PNP (0.54) PNPKDM4EMEN1ALDH1A1MAPT
SCHEMBL26155922 0.85 PNP (0.48) PNPKDM4EMEN1ALDH1A1MAPT
8-Aminoguanine SCHEMBL21761 0.85 PNP (1.00) PNPKDM4EMEN1ALDH1A1MAPT
SCHEMBL10597942 0.78 PNP (0.70) PNPKDM4EMEN1ALDH1A1MAPT
SCHEMBL3291323 0.76 NUDT1 (0.44) PNPKDM4EMEN1ALDH1A1MAPT
SCHEMBL843932 0.76 PNP (0.73) PNPKDM4EMEN1ALDH1A1MAPT
SCHEMBL20577 0.76 PNP (0.73) PNPKDM4EMEN1ALDH1A1MAPT
SCHEMBL844207 0.76 PNP (0.73) PNPKDM4EMEN1ALDH1A1MAPT
SCHEMBL6686388 0.76 PNP (0.73) PNPKDM4EMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6845 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106497-A2 FUNCTIONALIZED CIRCULAR RNA AND METHODS AND INTERMEDIATES FOR THEIR PRODUCTION SIEĆ BADAWCZA ŁUKASIEWICZ – PORT POLSKI OSRODEK ROZWOJU TECHNOLOGII (PL) 2026-05-21 WO claimed
WO-2026099790-A1 DEVICE USING ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2026-05-15 WO claimed
WO-2026099316-A1 COMPOUNDS AND METHODS FOR REDUCING ARHGEF6 EXPRESSION ASTRAZENECA AB (SE) 2026-05-15 WO claimed
US-20260131157-A1 METHODS OF USING ALTERNATING ELECTRIC FIELDS NOVOCURE GMBH (CH) 2026-05-14 US claimed
US-20260115161-A1 2-HYDROXY-OCTADECENE-9-CIS-OATE FOR USE IN THE TREATMENT OF ONCOLOGICAL PATHOLOGIES AND NEUROPATHIC PAIN LAMINAR PHARMACEUTICALS S A (ES) 2026-04-30 US claimed
US-12569572-B2 Messenger RNA therapy for the treatment of Friedreich's ataxia TRANSLATE BIO, INC. (US) 2026-03-10 US claimed
EP-4663187-A1 2-HYDROXY-OCTADECENE-9-CIS-OATE FOR USE IN THE TREATMENT OF ONCOLOGICAL PATHOLOGIES AND NEUROPATHIC PAIN Laminar Pharmaceuticals, S.A. (ES) 2025-12-17 EP claimed
EP-4452256-B1 METHODS OF TREATING BRAIN TUMOURS AND NEUROBLASTOMAS ASTRAZENECA AB (SE) 2025-12-10 EP claimed
US-12473663-B2 Compositions and methods for immune repertoiresequencing Life Technologies Corporation (US) 2025-11-18 US claimed
US-20250312347-A1 THERAPEUTIC BENEFIT OF SUBOPTIMALLY ADMINISTERED CHEMICAL COMPOUNDS BROWN DENNIS M (US) 2025-10-09 US claimed
US-5386030-A Chemical intermediates INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCE OF THE CZECH REPUBLIC (CZ) 1995-01-31 US claimed
EP-0630381-A4 ANTIVIRAL ACYCLIC PHOSPHONOMETHOXYALKYL SUBSTITUTED, ALKENYL AND ALKYNYL PURINE AND PYRIMIDINE DERIVATIVES. 1995-01-04 EP claimed
EP-0630381-A1 ANTIVIRAL ACYCLIC PHOSPHONOMETHOXYALKYL SUBSTITUTED, ALKENYL AND ALKYNYL PURINE AND PYRIMIDINE DERIVATIVES. ACAD OF SCIENCE CZECH REPUBLIC (CS) 1994-12-28 EP claimed
EP-0625985-A1 METHOD AND RING-OPENED PURINE COMPOUNDS FOR LABELING POLYNUCLEOTIDES. UNIV MIAMI (US) 1994-11-30 EP claimed
WO-1993011146-A1 METHOD AND RING-OPENED PURINE COMPOUNDS FOR LABELING POLYNUCLEOTIDES UNIVERSITY OF MIAMI (US) 1993-06-10 WO claimed
EP-0540693-A1 THE REDUCTION OF NON-SPECIFIC AMPLIFICATION DURING $i(IN VITRO) NUCLEIC ACID AMPLIFICATION USING MODIFIED NUCLEIC ACID BASES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1993-05-12 EP claimed
US-5208221-A Nucleotides and intermediates for herpes virus or leukemia virus BRISTOL-MYERS SQUIBB COMPANY (US) 1993-05-04 US claimed
WO-1993007157-A1 ANTIVIRAL ACYCLIC PHOSPHONOMETHOXYALKYL SUBSTITUTED, ALKENYL AND ALKYNYL PURINE AND PYRIMIDINE DERIVATIVES INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OFTHE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1993-04-15 WO claimed
WO-1992001814-A2 THE REDUCTION OF NON-SPECIFIC AMPLIFICATION DURING IN VITRO NUCLEIC ACID AMPLIFICATION USING MODIFIED NUCLEIC ACID BASES F. HOFFMANN-LA-ROCHE AG (CH) 1992-02-06 WO claimed
EP-0269947-A1 Antiviral phosphonomethoxyalkylene purine and pyrimidine derivatives INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CS) 1988-06-08 EP claimed