SCHEMBL42760

SCHEMBL42760

Nc1nc2nc(O)[nH]c2c(=O)[nH]1

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PNP P00491 5/20 0.73
FGFR1 P11362 1/20 0.56
FGFR2 P21802 1/20 0.56
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 1/20 0.53
MAPT P10636 1/20 0.53
THRB P10828 1/20 0.53
HPGD P15428 1/20 0.53
KMT2A Q03164 1/20 0.53
HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
8-Aminoguanine SCHEMBL5513824 0.98 PNP (0.77) PNPFGFR1FGFR2KDM4EMEN1
8-Aminoguanine SCHEMBL21761 0.85 PNP (1.00) PNPFGFR1FGFR2KDM4EMEN1
SCHEMBL19461404 0.80 PNP (0.47) PNPFGFR1FGFR2KDM4EMEN1
SCHEMBL22883 0.76 PNP (0.73) PNPFGFR1FGFR2KDM4EMEN1
SCHEMBL20577 0.76 PNP (0.73) PNPFGFR1FGFR2KDM4EMEN1
SCHEMBL843932 0.76 PNP (0.73) PNPFGFR1FGFR2KDM4EMEN1
SCHEMBL844207 0.76 PNP (0.73) PNPFGFR1FGFR2KDM4EMEN1
SCHEMBL9116 0.76 PNP (0.73) PNPFGFR1FGFR2KDM4EMEN1
SCHEMBL6686388 0.76 PNP (0.73) PNPFGFR1FGFR2KDM4EMEN1
SCHEMBL2051361 0.76 PNP (0.73) PNPFGFR1FGFR2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5482 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12630827-B2 Antisense oligonucleotides targeting SCN2A for the treatment of SCN1A encephalopathies ROGCON, INC. (US) 2026-05-19 US claimed
US-20250295658-A1 ANTIPARASITIC AGENTS AND METHODS WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH 2025-09-25 US claimed
US-20250257360-A1 OLIGONUCLEOTIDE INTERFERENCE TREATMENTS OF PROSTATE CANCER UNIV OKLAHOMA (US) 2025-08-14 US claimed
CN-113151261-B Antisense oligonucleotides as inhibitors of TGF-R signaling 神经视觉医药有限公司 2025-06-17 CN claimed
US-20250179503-A1 METHODS OF USING OLIGOMERIC COMPOUNDS TO TREAT SCN2A-RELATED DISORDERS PRAXIS PREC MEDICINES INC (US) 2025-06-05 US claimed
US-20250146073-A1 METHODS FOR THE TREATMENT OF SCN2A-RELATED DISORDERS PRAXIS PREC MEDICINES INC (US) 2025-05-08 US claimed
EP-4549577-A1 NOVEL INDUCED CYTOPLASMIC IVT (ICIVT)-LIKE COMPOSITION AND THE RELATED VACCINE MEDICINE DESIGNS THEREOF Mello Biotech Taiwan Co., Ltd. (TW) 2025-05-07 EP claimed
US-20250115932-A1 INDUCED CYTOPLASMIC IVT (ICIVT)-LIKE COMPOSITION AND THE RELATED VACCINE MEDICINE DESIGNS THEREOF MELLO BIOTECH TAIWAN CO., LTD. (TW) 2025-04-10 US claimed
EP-4506456-A1 NOVEL OXO-RNA COMPOSITIONS AND THE RELATED APPLICATIONS THEREOF Lin, Shi-Lung (US) 2025-02-12 EP claimed
EP-4504945-A2 OLIGONUCLEOTIDE INTERFERENCE TREATMENTS OF PROSTATE CANCER The Board of Regents of the University of Oklahoma (US) 2025-02-12 EP claimed
US-5552285-A DIAGNOSIS AND MONITORING OF INFLAMMATORY AND AUTOIMMUNE DISEASES NEW YORK UNIVERSITY (US) 1996-09-03 US claimed
EP-0706581-A1 DNA PROFILES AS AN INDICATOR OF CELLULAR REDOX POTENTIAL AND CANCER RISK PACIFIC NORTHWEST RESEARCH FOUNDATION (US) 1996-04-17 EP claimed
US-5386030-A Chemical intermediates INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCE OF THE CZECH REPUBLIC (CZ) 1995-01-31 US claimed
EP-0630381-A4 ANTIVIRAL ACYCLIC PHOSPHONOMETHOXYALKYL SUBSTITUTED, ALKENYL AND ALKYNYL PURINE AND PYRIMIDINE DERIVATIVES. 1995-01-04 EP claimed
EP-0630381-A1 ANTIVIRAL ACYCLIC PHOSPHONOMETHOXYALKYL SUBSTITUTED, ALKENYL AND ALKYNYL PURINE AND PYRIMIDINE DERIVATIVES. ACAD OF SCIENCE CZECH REPUBLIC (CS) 1994-12-28 EP claimed
WO-1994025626-A1 DNA PROFILES AS AN INDICATOR OF CELLULAR REDOX POTENTIAL AND CANCER RISK PACIFIC NORTHWEST RESEARCH FOUNDATION (US) 1994-11-10 WO claimed
US-5208221-A Nucleotides and intermediates for herpes virus or leukemia virus BRISTOL-MYERS SQUIBB COMPANY (US) 1993-05-04 US claimed
WO-1993007157-A1 ANTIVIRAL ACYCLIC PHOSPHONOMETHOXYALKYL SUBSTITUTED, ALKENYL AND ALKYNYL PURINE AND PYRIMIDINE DERIVATIVES INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OFTHE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1993-04-15 WO claimed
WO-1992015707-A1 IMMUNOASSAY FOR ANTIBODIES TO OXIDIZED DNA AND USES THEREOF NEW YORK UNIVERSITY (US) 1992-09-17 WO claimed
EP-0269947-A1 Antiviral phosphonomethoxyalkylene purine and pyrimidine derivatives INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CS) 1988-06-08 EP claimed