SCHEMBL22894540

SCHEMBL22894540

CN1CCN(c2ccc(Br)cc2Cl)C1=O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.39
SLC22A12 Q96S37 1/20 0.37
SRD5A1 P18405 1/20 0.37
KDM4E B2RXH2 2/20 0.36
MAPT P10636 1/20 0.36
RAD52 P43351 1/20 0.36
KMT2A Q03164 1/20 0.36
BRD4 O60885 1/20 0.36
CASP2 P42575 1/20 0.35
BCL2A1 Q16548 1/20 0.35
CRHR1 P34998 1/20 0.35
SCN9A Q15858 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22894543 0.83 MEN1 (0.46) P2RX7SRD5A1MAPTKMT2ABRD4
SCHEMBL30931056 0.83 MEN1 (0.46) P2RX7SRD5A1MAPTKMT2ABRD4
SCHEMBL22894546 0.81 SCN9A (0.42) P2RX7SRD5A1KDM4EMAPTBRD4
SCHEMBL22894548 0.80 SMN1; SMN2 (0.49) P2RX7SRD5A1KDM4EMAPTKMT2A
SCHEMBL29182733 0.80 SLC22A12 (0.42) P2RX7SLC22A12MAPTKMT2ACASP2
SCHEMBL27389435 0.79 PTGS1 (0.42) P2RX7KDM4EMAPTRAD52SCN9A
SCHEMBL17907336 0.75 CYP2D6 (0.48) P2RX7SLC22A12KDM4EMAPTKMT2A
SCHEMBL16531977 0.75 P2RX7 (0.42) P2RX7SLC22A12
SCHEMBL24719734 0.73 HSD17B10 (0.46) SLC22A12SRD5A1KDM4EKMT2ATSHR
SCHEMBL16531970 0.73 GLA (0.39) P2RX7SLC22A12SRD5A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3042907-B1 DGAT1 INHIBITOR AND PREPARATION METHOD AND USE THEREOF QUINGDAO HUANGHAI PHARMACEUTICAL CO LTD (CN) 2021-01-13 EP disclosed