SCHEMBL22894546

SCHEMBL22894546

CN1CCN(c2ccc(Br)cc2F)C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.42
SCN10A Q9Y5Y9 1/20 0.42
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA5A P35218 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA13 Q8N1Q1 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
PARP1 P09874 1/20 0.40
CCR1 P32246 2/20 0.38
CCR2 P41597 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
ALDH1A1 P00352 4/20 0.37
HPGD P15428 2/20 0.37
TSHR P16473 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29348971 0.91 CCR1 (0.39) SCN9ASCN10ACA12CA1CA2
SCHEMBL8302887 0.84 CA12 (0.55) SCN9ASCN10ACA12CA1CA2
SCHEMBL30931056 0.83 MEN1 (0.46) SCN9ASCN10APARP1ALDH1A1HPGD
SCHEMBL22894543 0.83 MEN1 (0.46) SCN9ASCN10APARP1ALDH1A1HPGD
SCHEMBL22542026 0.83 SCN9A (0.43) SCN9ASCN10ACA12CA1CA2
SCHEMBL22894540 0.81 P2RX7 (0.39) SCN9ASCN10ATSHRMAPTSRD5A1
SCHEMBL22894548 0.80 SMN1; SMN2 (0.49) SCN9ASCN10APARP1ALDH1A1HPGD
SCHEMBL24478480 0.79 PARP1 (0.46) SCN9ASCN10ACA12CA1CA2
SCHEMBL24451807 0.79 SCN9A (0.41) SCN9ASCN10ACA12CA1CA2
SCHEMBL30931022 0.79 SCN9A (0.36) SCN9ASCN10APARP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022261204-A1 ANTICANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-12-15 WO disclosed
EP-3042907-B1 DGAT1 INHIBITOR AND PREPARATION METHOD AND USE THEREOF QUINGDAO HUANGHAI PHARMACEUTICAL CO LTD (CN) 2021-01-13 EP disclosed