SCHEMBL22894548

SCHEMBL22894548

CCc1cc(Br)ccc1N1CCN(C)C1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.49
TSHR P16473 2/20 0.49
LMNA P02545 1/20 0.49
HPGD P15428 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CRHR1 P34998 1/20 0.38
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
SRD5A1 P18405 1/20 0.36
P2RX7 Q99572 2/20 0.36
BRD4 O60885 1/20 0.35
CASP2 P42575 1/20 0.35
TP53 P04637 2/20 0.34
MAPT P10636 2/20 0.34
PARP1 P09874 1/20 0.34
SCN9A Q15858 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22894543 0.81 MEN1 (0.46) TSHRLMNAHPGDCRHR1ALDH1A1
SCHEMBL30931056 0.81 MEN1 (0.46) TSHRLMNAHPGDCRHR1ALDH1A1
SCHEMBL22894546 0.80 SCN9A (0.42) TSHRHPGDL3MBTL1ALDH1A1KDM4E
SCHEMBL22894540 0.80 P2RX7 (0.39) TSHRCRHR1KDM4ESRD5A1P2RX7
SCHEMBL18065422 0.78 LMNA (0.43) SMN1; SMN2TSHRLMNAHPGDL3MBTL1
SCHEMBL14864862 0.77 ALDH1A1 (0.43) SMN1; SMN2LMNAL3MBTL1ALDH1A1POLB
SCHEMBL17907343 0.76 SMN1; SMN2 (0.52) SMN1; SMN2TSHRLMNAHPGDL3MBTL1
SCHEMBL24196400 0.75 PARP1 (0.38) P2RX7BRD4PARP1SCN9ASCN10A
SCHEMBL22894471 0.75 TP53 (0.32) SMN1; SMN2TSHRLMNAHPGDL3MBTL1
SCHEMBL17907285 0.74 LMNA (0.40) SMN1; SMN2TSHRLMNAHPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3042907-B1 DGAT1 INHIBITOR AND PREPARATION METHOD AND USE THEREOF QUINGDAO HUANGHAI PHARMACEUTICAL CO LTD (CN) 2021-01-13 EP disclosed