SCHEMBL22908403

SCHEMBL22908403

COc1cc(-c2ccc(C#N)cn2)cc(Cl)c1C1C(=O)CC2(CCN(C(=O)c3ccccc3)CC2)CC1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.43
MAPK7 Q13164 1/20 0.41
USP2 O75604 4/20 0.40
TSHR P16473 4/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
AR P10275 1/20 0.40
CYP3A4 P08684 6/20 0.39
CYP2D6 P10635 2/20 0.39
FFAR2 O15552 1/20 0.39
ALDH1A1 P00352 2/20 0.38
PTGER4 P35408 1/20 0.38
PTGER2 P43116 1/20 0.38
PTGDR Q13258 1/20 0.38
MAPK1 P28482 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CCR8 P51685 2/20 0.36
KCNH2 Q12809 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22908434 0.90 IGF1R (0.39) MAPK7TSHRCYP1A2CYP2C9CYP3A4
SCHEMBL22908404 0.88 CHEK1 (0.36) GRM5MAPK7SMN1; SMN2CYP3A4FFAR2
SCHEMBL21361301 0.86 GRM5 (0.45) GRM5SMN1; SMN2ARCYP3A4CYP2D6
SCHEMBL21361292 0.84 TSHR (0.40) MAPK7TSHRCYP1A2CYP2C9CYP2D6
SCHEMBL24120370 0.84 GRM5 (0.42) GRM5MAPK7USP2TSHRCYP3A4
SCHEMBL22908402 0.83 CYP2D6 (0.42) USP2TSHRCYP1A2SMN1; SMN2CYP3A4
SCHEMBL21361307 0.81 CYP1A2 (0.38) MAPK7TSHRCYP1A2CYP2C9CYP2D6
SCHEMBL22908414 0.80 CYP1A2 (0.41) GRM5TSHRCYP1A2CYP2C9CYP3A4
SCHEMBL22908406 0.80 CYP2D6 (0.45) USP2TSHRCYP1A2CYP2C9SMN1; SMN2
SCHEMBL22908538 0.79 CCR8 (0.41) USP2TSHRCYP1A2CYP2C9SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021009048-A1 HERBICIDAL CYCLOHEXANEDIONE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2021-01-21 WO disclosed