SCHEMBL22908402

SCHEMBL22908402

COc1cc(-c2ncc(F)cn2)cc(Cl)c1C1C(=O)CC2(CCN(C(=O)c3ccccc3)CC2)CC1=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.42
HTR1A P08908 4/20 0.41
ALDH1A1 P00352 4/20 0.41
DRD2 P14416 3/20 0.41
ADRA1A P35348 3/20 0.41
CCR8 P51685 3/20 0.39
KCNH2 Q12809 3/20 0.39
CYP3A4 P08684 5/20 0.39
TSHR P16473 3/20 0.39
TNF P01375 1/20 0.39
LITAF Q99732 1/20 0.39
CYP1A2 P05177 3/20 0.39
MAPK1 P28482 2/20 0.38
USP2 O75604 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HSD17B10 Q99714 1/20 0.38
LRRK2 Q5S007 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22908406 0.89 CYP2D6 (0.45) CYP2D6HTR1AALDH1A1DRD2ADRA1A
SCHEMBL21361251 0.86 CYP3A4 (0.42) CYP2D6HTR1AALDH1A1CYP3A4TSHR
SCHEMBL22908403 0.83 GRM5 (0.43) CYP2D6HTR1AALDH1A1DRD2ADRA1A
SCHEMBL22859575 0.82 CYP2D6 (0.37) CYP2D6ALDH1A1TSHRCYP1A2MEN1
SCHEMBL24120123 0.82 ALDH1A1 (0.36) CYP2D6ALDH1A1KCNH2CYP3A4CYP1A2
SCHEMBL22908538 0.79 CCR8 (0.41) CYP2D6HTR1AALDH1A1DRD2ADRA1A
SCHEMBL21361271 0.79 CYP2D6 (0.46) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL21361309 0.79 CYP2D6 (0.35) CYP2D6ALDH1A1TSHRCYP1A2MEN1
SCHEMBL21361218 0.77 ACACB (0.34) TNFLITAF
SCHEMBL21361247 0.76 L3MBTL1 (0.42) CYP2D6ALDH1A1CCR8KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021009048-A1 HERBICIDAL CYCLOHEXANEDIONE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2021-01-21 WO disclosed