SCHEMBL22908985

SCHEMBL22908985

CCOC(=O)c1sc2cccc(Br)c2c1CBr

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
KDM4E B2RXH2 4/20 0.53
L3MBTL1 Q9Y468 3/20 0.53
GAA P10253 2/20 0.53
TSHR P16473 2/20 0.53
HPGD P15428 2/20 0.53
HSD17B10 Q99714 2/20 0.53
GLA P06280 1/20 0.53
MAPK1 P28482 1/20 0.53
LMNA P02545 3/20 0.44
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
RXFP1 Q9HBX9 2/20 0.44
KMT2A Q03164 4/20 0.43
MAPT P10636 5/20 0.42
NPSR1 Q6W5P4 1/20 0.42
NOD2 Q9HC29 1/20 0.42
MEN1 O00255 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29443017 0.86 ALDH1A1 (0.69) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL22905016 0.86 ALDH1A1 (0.69) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL23112012 0.86 ALDH1A1 (0.69) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL22909023 0.85 ALDH1A1 (0.56) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL22908996 0.85 ALDH1A1 (0.51) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL30765073 0.85 ALDH1A1 (0.51) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL22909057 0.85 MAPT (0.54) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL29513197 0.85 MAPT (0.54) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL22908998 0.83 ALDH1A1 (0.52) ALDH1A1KDM4EL3MBTL1GAATSHR
SCHEMBL23112085 0.83 ALDH1A1 (0.49) ALDH1A1KDM4EL3MBTL1GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250092009-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING CTXT PTY LTD (AU) 2025-03-20 US disclosed
CN-114206882-B Benzothiophene, thienopyridine and thienopyrimidine derivatives for modulating STING CTXT私人有限公司 2024-11-12 CN disclosed
CN-112424181-B Substituted condensed thiophenes as STING modulators 希泰克斯特私人有限公司 2024-02-27 CN disclosed
EP-3793988-B1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING CTXT PTY LTD (AU) 2023-11-15 EP disclosed
EP-3793988-B1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING CTXT PTY LTD (AU) 2023-11-15 EP disclosed
EP-3999185-B1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LTD (AU) 2023-08-30 EP disclosed
US-20230227423-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING CTXT PTY LTD (AU) 2023-07-20 US disclosed
US-20230227423-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING CTXT PTY LTD (AU) 2023-07-20 US disclosed
US-20230227423-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING CTXT PTY LTD (AU) 2023-07-20 US disclosed
US-11613525-B2 Substituted condensed thiophenes as modulators of sting CTXT PTY LIMITED (AU) 2023-03-28 US disclosed
US-20220389032-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LTD. (AU) 2022-12-08 US disclosed
US-20210214333-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING CTXT PTY LTD. (AU) 2021-07-15 US disclosed
EP-3793988-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING Ctxt Pty Ltd (AU) 2021-03-24 EP disclosed
CN-112424181-A Substituted condensed thiophenes as STING modulators 希泰克斯特私人有限公司 2021-02-26 CN disclosed
WO-2021009365-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LIMITED (AU) 2021-01-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230227423-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING STING1, CGAS, IRF3 ALDH1A1 4660/4885KDM4E 1469/4885L3MBTL1 938/4885
US-20210214333-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING STING1, CGAS, IRF3 ALDH1A1 4719/4885KDM4E 1519/4885L3MBTL1 983/4885
US-20220389032-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING STING1, CGAS, MAVS ALDH1A1 3516/4885KDM4E 1256/4885L3MBTL1 2546/4885
US-11613525-B2 Substituted condensed thiophenes as modulators of sting STING1, CGAS, IRF3 ALDH1A1 4719/4885KDM4E 1519/4885L3MBTL1 983/4885
US-20250092009-A1 SUBSTITUTED CONDENSED THIOPHENES AS MODULATORS OF STING STING1, CGAS, IRF3 ALDH1A1 4660/4885KDM4E 1469/4885L3MBTL1 938/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.