SCHEMBL22908993

SCHEMBL22908993

CCOC(=O)c1sc2ccnc(OC)c2c1C=O

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.49
CDC7 O00311 10/20 0.48
DBF4 Q9UBU7 10/20 0.48
KDM4E B2RXH2 5/20 0.45
LMNA P02545 4/20 0.45
ALDH1A1 P00352 3/20 0.45
CASP1 P29466 1/20 0.41
HTT P42858 1/20 0.41
CASP7 P55210 1/20 0.41
GAA P10253 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
GLA P06280 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
STING1 Q86WV6 1/20 0.41
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29513312 1.00 HSD17B10 (0.49) HSD17B10CDC7DBF4KDM4ELMNA
SCHEMBL29693859 0.85 HSD17B10 (0.63) HSD17B10CDC7DBF4KDM4ELMNA
SCHEMBL22905056 0.85 HSD17B10 (0.63) HSD17B10CDC7DBF4KDM4ELMNA
SCHEMBL22909082 0.84 STING1 (0.49) HSD17B10CDC7DBF4KDM4ELMNA
SCHEMBL22908994 0.81 HSD17B10 (0.49) HSD17B10CDC7DBF4KDM4ELMNA
SCHEMBL30765125 0.81 HSD17B10 (0.49) HSD17B10CDC7DBF4KDM4ELMNA
SCHEMBL29513181 0.78 ALDH1A1 (0.51) HSD17B10KDM4ELMNAALDH1A1HTT
SCHEMBL22909058 0.78 ALDH1A1 (0.51) HSD17B10KDM4ELMNAALDH1A1HTT
SCHEMBL22904903 0.77 HSD17B10 (0.47) HSD17B10CDC7DBF4KDM4ELMNA
SCHEMBL29443064 0.77 HSD17B10 (0.47) HSD17B10CDC7DBF4KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12384801-B2 Benzothiophene, thienopyridine and thienopyrimidine derivatives for the modulation of sting CTXT PTY LTD. (AU) 2025-08-12 US disclosed
EP-3999185-B1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LTD (AU) 2023-08-30 EP disclosed
EP-3999185-B1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LTD (AU) 2023-08-30 EP disclosed
US-20220389032-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LTD. (AU) 2022-12-08 US disclosed
US-20220389032-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LTD. (AU) 2022-12-08 US disclosed
EP-3999185-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT Pty Limited (AU) 2022-05-25 EP disclosed
CN-114206882-A Benzothiophene, thienopyridine, and thienopyrimidine derivatives for modulation of STING CTXT私人有限公司 2022-03-18 CN disclosed
WO-2021009365-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LIMITED (AU) 2021-01-21 WO disclosed
WO-2021009365-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING CTXT PTY LIMITED (AU) 2021-01-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12384801-B2 Benzothiophene, thienopyridine and thienopyrimidine derivatives for the modulation of sting STING1, CGAS, MAVS HSD17B10 4526/4885CDC7 2787/4885DBF4 175/4885
US-20220389032-A1 BENZOTHIOPHENE, THIENOPYRIDINE AND THIENOPYRIMIDINE DERIVATIVES FOR THE MODULATION OF STING STING1, CGAS, MAVS HSD17B10 4526/4885CDC7 2787/4885DBF4 175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.