SCHEMBL22914964

SCHEMBL22914964

Cc1ccc(Cl)cc1NC(O)c1cn(-c2cc(O)ccc2F)nn1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RXRA P19793 5/20 0.34
GRIN1 Q05586 5/20 0.34
GRIN2B Q13224 5/20 0.34
NOTUM Q6P988 3/20 0.34
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.32
AGPAT2 O15120 1/20 0.31
MAPT P10636 1/20 0.31
ATM Q13315 1/20 0.31
P2RX7 Q99572 1/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22914939 0.78 MAPT (0.48) MAPTUSP2
SCHEMBL5128529 0.73 NOTUM (0.54) RXRAGRIN1GRIN2BNOTUMCYP1A2
SCHEMBL22914931 0.65 MAPT (0.48) NOTUMMAPTUSP2
SCHEMBL29709808 0.65 MAPT (0.48) NOTUMMAPTUSP2
SCHEMBL16982958 0.65 NOTUM (0.39) RXRAGRIN1GRIN2BNOTUMCYP1A2
SCHEMBL16983100 0.64 RXRA (0.42) RXRAGRIN1GRIN2BNOTUMCYP3A4
SCHEMBL5126332 0.64 CYP3A4 (0.39) RXRAGRIN1GRIN2BNOTUMCYP1A2
SCHEMBL22914920 0.62 MAPT (0.50) MAPTUSP2
SCHEMBL29709838 0.62 MAPT (0.50) MAPTUSP2
SCHEMBL5483071 0.62 NR1I2 (0.37) RXRAGRIN1GRIN2BNOTUMCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021016594-A1 SECOND GENERATION INHIBITORS OF MITOCHONDRIAL PERMEABILITY TRANSITION PORE WITH IMPROVED PLASMA STABILITY OREGON HEALTH & SCIENCE UNIVERSITY (US) 2021-01-28 WO disclosed