SCHEMBL2292207

SCHEMBL2292207

Cc1cccc(CNC(=O)CON=C2CCN(S(=O)(=O)c3cccc(C(F)(F)F)c3)CC2)c1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 2/20 0.45
MAPT P10636 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 1/20 0.43
PLA2G1B P04054 1/20 0.43
PKM P14618 1/20 0.43
ATG4B Q9Y4P1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2297393 0.91 LMNA (0.52) KMT2AMEN1GAALMNAPLA2G1B
SCHEMBL2290518 0.91 KMT2A (0.47) KMT2AMEN1GAAMAPTLMNA
SCHEMBL2291401 0.90 KMT2A (0.51) KMT2AGAAL3MBTL1LMNAPKM
SCHEMBL3640385 0.90 LMNA (0.42) KMT2AMEN1LMNA
SCHEMBL2291154 0.88 MEN1 (0.50) KMT2AMEN1GAAMAPTLMNA
SCHEMBL2295296 0.87 NAMPT (0.48) KMT2AMEN1GAALMNA
SCHEMBL2293920 0.87 NAMPT (0.51) KMT2AMEN1LMNA
SCHEMBL2292597 0.87 KMT2A (0.46) KMT2AMEN1GAAMAPTL3MBTL1
SCHEMBL2296261 0.85 PKM (0.47) KMT2AMEN1GAAMAPTLMNA
SCHEMBL2296022 0.85 KMT2A (0.45) KMT2AMEN1GAAMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110190300-A1 AMIDE COMPOUNDS AND THE USE THEREOF EURO-CELTIQUE S.A. (LU) 2011-08-04 US disclosed
US-20110190300-A1 AMIDE COMPOUNDS AND THE USE THEREOF EURO-CELTIQUE S.A. (LU) 2011-08-04 US disclosed
US-20110190300-A1 AMIDE COMPOUNDS AND THE USE THEREOF EURO-CELTIQUE S.A. (LU) 2011-08-04 US disclosed
EP-2164326-A1 AMIDE COMPOUNDS AND THE USE THEREOF Euro-Celtique, S.A. (LU) 2010-03-24 EP disclosed
WO-2008150447-A1 AMIDE COMPOUNDS AND THE USE THEREOF EURO-CELTIQUE S.A. (LU) 2008-12-11 WO disclosed
WO-2008150447-A1 AMIDE COMPOUNDS AND THE USE THEREOF EURO-CELTIQUE S.A. (LU) 2008-12-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110190300-A1 AMIDE COMPOUNDS AND THE USE THEREOF CACNA1E, CACNA1B, CACNA1S KMT2A 2564/4885MEN1 3484/4885GAA 3413/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.