SCHEMBL22930892

SCHEMBL22930892

N#CCC(N)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.38
KCNA5 P22460 1/20 0.38
KCNH2 Q12809 1/20 0.38
GPR139 Q6DWJ6 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
CETP P11597 1/20 0.37
KIF11 P52732 1/20 0.37
SLC6A2 P23975 5/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22952674 1.00 ADORA2A (0.38) ADORA2AADORA1TRPM8KCNA5KCNH2
Hydrochloric Acid SCHEMBL28719364 0.99 SLC6A2 (0.38) ADORA2AADORA1TRPM8KCNA5KCNH2
Hydrochloric Acid SCHEMBL28719366 0.99 SLC6A2 (0.38) ADORA2AADORA1TRPM8KCNA5KCNH2
SCHEMBL22952726 0.86 ADORA2A (0.37) ADORA2AADORA1TRPM8KCNA5KCNH2
Hydrochloric Acid SCHEMBL28715423 0.85 SLC6A2 (0.36) ADORA2AADORA1TRPM8KCNA5KCNH2
Hydrochloric Acid SCHEMBL28715421 0.85 SLC6A2 (0.36) ADORA2AADORA1TRPM8KCNA5KCNH2
SCHEMBL18704160 0.82 CETP (0.43) GPR139CETPSLC6A2
SCHEMBL171242 0.82 GPR139 (0.43) KCNA5KCNH2GPR139CTSSCTSK
SCHEMBL734938 0.81 KIF11 (0.43) TRPM8CETPKIF11SLC6A2
SCHEMBL16563768 0.81 PDE2A (0.40) SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461327-A Spiro urea derivatives 爱杜西亚药品有限公司 2022-12-09 CN disclosed
EP-3466953-B1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVE AS JANUS KINASE INHIBITOR INCYTE HOLDINGS CORP (US) 2021-02-03 EP disclosed