SCHEMBL2293486

SCHEMBL2293486

NC(=O)c1ncc2ccccc2c1O

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.49
EGLN1 Q9GZT9 3/20 0.47
PIM1 P11309 1/20 0.42
KDM4E B2RXH2 2/20 0.41
GPR3 P46089 1/20 0.41
LCK P06239 2/20 0.41
MAP2K3 P46734 1/20 0.41
MAP2K6 P52564 1/20 0.41
BTK Q06187 1/20 0.41
MAP3K19 Q56UN5 1/20 0.41
NEK10 Q6ZWH5 1/20 0.41
LDHA P00338 1/20 0.41
ILK Q13418 1/20 0.38
PTPN22 Q9Y2R2 1/20 0.38
IKBKB O14920 1/20 0.38
EGLN2 Q96KS0 3/20 0.38
HTT P42858 1/20 0.37
ELANE P08246 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8150746 0.84 LDHA (0.50) MAOAEGLN1KDM4EGPR3LDHA
SCHEMBL5141974 0.80 EGLN2 (0.47) EGLN1MAP2K3IKBKBEGLN2
SCHEMBL28007224 0.78 MAOA (0.52) MAOAEGLN1KDM4ELCKHTT
SCHEMBL15631107 0.78 MAOA (0.49) MAOAEGLN1KDM4EGPR3LDHA
SCHEMBL30394217 0.77 EGLN1 (0.67) EGLN1EGLN2
SCHEMBL6789839 0.76 KDM4E (0.44) EGLN1KDM4ELCKMAP2K3MAP2K6
SCHEMBL1342390 0.76 FEN1 (0.56) EGLN1PIM1KDM4EHTT
SCHEMBL27755791 0.76 PDE4B (0.46) EGLN1EGLN2
SCHEMBL31501044 0.73 EGLN1 (0.68) EGLN1EGLN2
SCHEMBL821293 0.73 EGLN1 (0.68) EGLN1EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960363-B1 QUINOLONE BASED COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS AND USES THEREOF AMGEN INC (US) 2014-01-22 EP disclosed
US-20110263642-A1 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS FIBROGEN, INC. (US) 2011-10-27 US disclosed
EP-2341904-A1 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS Fibrogen, Inc. (US) 2011-07-13 EP disclosed
WO-2010024908-A1 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS FIBROGEN, INC. (US) 2010-03-04 WO disclosed
WO-2010024911-A1 METHODS FOR INCREASING NEUROGENESIS FIBROGEN, INC. (US) 2010-03-04 WO disclosed
US-20040180910-A1 Heterocycle carboxamides as antiviral agents SCHNUTE MARK E (US) 2004-09-16 US disclosed
US-6730682-B2 HERPES VIRUS PHARMACIA & UPJOHN COMPANY 2004-05-04 US disclosed
EP-1363907-A2 HETEROCYCLE CARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2003-11-26 EP disclosed
US-20020019397-A1 Heterocycle carboxamides as antiviral agents PHARMACIA & UPJOHN COMPANY 2002-02-14 US disclosed
WO-2002004443-A2 HETEROCYCLE CARBOXAMIDES AS ANTIVIRAL AGENTS PHARMACIA & UPJOHN COMPANY (US) 2002-01-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040180910-A1 Heterocycle carboxamides as antiviral agents ZC3HAV1, ZC3HAV1L, HDAC1 MAOA 2284/4885EGLN1 134/4885PIM1 589/4885
US-20020019397-A1 Heterocycle carboxamides as antiviral agents ZC3HAV1, ZC3HAV1L, HDAC1 MAOA 2284/4885EGLN1 134/4885PIM1 589/4885
US-20110263642-A1 METHODS FOR TREATMENT OF MULTIPLE SCLEROSIS PMP22, MAG, NEFM MAOA 1659/4885EGLN1 2695/4885PIM1 4403/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.