SCHEMBL2294879

SCHEMBL2294879

O=C(OC(Cl)C(Cl)(Cl)Cl)OC(Cl)C(Cl)(Cl)Cl

nearest known ligand 0.30

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4349836 0.81 ELANE (0.32)
SCHEMBL1502043 0.80
SCHEMBL2294883 0.80 ALDH1A1 (0.33) LMNA
Hydrochloric Acid SCHEMBL11629040 0.78 LMNA (0.32) LMNA
SCHEMBL7940239 0.78
SCHEMBL20118113 0.78 TSHR (0.43) LMNA
SCHEMBL29001764 0.78
SCHEMBL10898329 0.76
SCHEMBL10455575 0.76
SCHEMBL11592647 0.76 HCAR2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364159-A1 DEUTERATED MACROCYCLIC INHIBITORS OF VIRAL NS3 PROTEASE CONCERT PHARMACEUTICALS, INC. (US) 2011-09-14 EP disclosed
US-20110196012-A1 DEUTERATED MACROCYCLIC INHIBITORS OF VIRAL NS3 PROTEASE CONCERT PHARMACEUTICALS, INC. (US) 2011-08-11 US disclosed
WO-2010048468-A1 DEUTERATED MACROCYCLIC INHIBITORS OF VIRAL NS3 PROTEASE CONCERT PHARMACEUTICALS, INC. (US) 2010-04-29 WO disclosed
US-6444825-B1 CHEMICAL INTERMEDIATE FOR TAXOL AVENTIS PHARMA S.A. (FR) 2002-09-03 US disclosed
US-6043375-A Process for the preparation of an oxazolidinecarboxylic acid which is useful for preparing therapeutically active taxoids RHONE-POULENC RORER S.A. (FR) 2000-03-28 US disclosed
US-4960881-A REACTING AMINO ACID WITH ALPHA-CHLORINATED CARBONATE IN SOLVENT IN PRESENCE OF ACID SCAVENGER SOCIETE NATIONALE DES POUDRES ET EXPLOSIFS (FR) 1990-10-02 US disclosed
US-4652665-A BLOCK AMINE FUNCTION OF AMINO ACIDS; PEPTIDE SYNTHESIS SOCIETE NATIONALE DES POUDRES ET EXPLOSIFS (FR) 1987-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110196012-A1 DEUTERATED MACROCYCLIC INHIBITORS OF VIRAL NS3 PROTEASE DPP3, SPINT2, DPP4 LMNA 2871/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.