SCHEMBL22952989

SCHEMBL22952989

Cc1cc(O)c2c3c1Cc1c(ccc(O)c1O)C3CNC2

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.43
KIF11 P52732 1/20 0.39
HTR2A P28223 1/20 0.33
MAPK1 P28482 2/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
THPO P40225 1/20 0.33
HSD17B10 Q99714 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
PMP22 Q01453 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22952985 0.82 PARP1 (0.32) PARP1KIF11
SCHEMBL22952988 0.82 DRD1 (0.33) PARP1KIF11MAPK1CYP3A4TSHR
SCHEMBL22952984 0.82 DRD2 (0.32) PARP1KIF11HTR2A
SCHEMBL22952987 0.80 PARP1 (0.41) PARP1KIF11HTR2AMAPK1CYP3A4
SCHEMBL22953386 0.80 PARP1 (0.39) PARP1KIF11HTR2ALMNA
SCHEMBL22953343 0.78 PARP1 (0.41) PARP1KIF11MAPK1CYP3A4ALOX15
SCHEMBL22952986 0.77 PARP1 (0.46) PARP1KIF11HTR2AMAPK1CYP3A4
SCHEMBL18309835 0.75 PARP1 (0.59) PARP1KIF11MAPK1CYP3A4ALOX15
SCHEMBL22953390 0.74 HTR2A (0.36) PARP1KIF11HTR2A
SCHEMBL16938669 0.73 HTR2A (0.60) PARP1KIF11HTR2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021021922-A1 COMPOUNDS AND METHODS FOR TREATING FIBROTIC PATHOLOGIES MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2021-02-04 WO disclosed