SCHEMBL22965739

SCHEMBL22965739

NNc1cc(Cl)cc(Br)c1N

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
CA9 Q16790 3/20 0.34
TP53 P04637 1/20 0.33
CYP3A4 P08684 1/20 0.33
CA3 P07451 1/20 0.31
ERN1 O75460 1/20 0.31
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25167009 0.81 GAA (0.36) GAAMAPTCA1CA2CA9
SCHEMBL31220169 0.81 GAA (0.36) GAAMAPTCA1CA2CA9
SCHEMBL1639812 0.78 GAA (0.58) GAAMAPTCA1CA2CA9
SCHEMBL16352569 0.75 GAA (0.51) GAAMAPTCYP3A4
SCHEMBL22965725 0.74 GAA (0.40) GAAMAPTCA1CA2CA9
SCHEMBL25292899 0.72 ALDH1A1 (0.32) MAPT
SCHEMBL7042377 0.72 CA2 (0.39) GAAMAPTCA1CA2
SCHEMBL31050390 0.72 CA1 (0.54) GAAMAPTCA1CA2CA9
SCHEMBL18421429 0.72 TSHR (0.35) GAATP53CYP3A4ERN1MCL1
SCHEMBL3605101 0.72 CA1 (0.54) GAAMAPTCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021026375-A1 FUSED BICYCLIC COMPOUNDS FOR THE TREATMENT OF PAIN ALKERMES, INC. (US) 2021-02-11 WO disclosed