SCHEMBL22966699

SCHEMBL22966699

CC(=O)Oc1c(O)c(O)cc2oc(-c3ccccc3)cc(=O)c12

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREB1 P16220 6/20 0.82
ABCB1 P08183 9/20 0.66
CYP3A4 P08684 4/20 0.66
MAPT P10636 4/20 0.66
CYP2C9 P11712 3/20 0.66
CYP2C19 P33261 3/20 0.66
MEN1 O00255 3/20 0.66
ALDH1A1 P00352 3/20 0.66
CYP1A1 P04798 3/20 0.66
CYP1A2 P05177 3/20 0.66
KMT2A Q03164 3/20 0.66
SMN1; SMN2 Q16637 3/20 0.66
CYP1B1 Q16678 3/20 0.66
FTO Q9C0B1 3/20 0.66
PRSS1 P07477 2/20 0.66
PRSS2 P07478 2/20 0.66
PRSS3 P35030 2/20 0.66
PTPRS Q13332 2/20 0.66
KDM4E B2RXH2 2/20 0.66
GABRP O00591 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29008532 0.93 CREB1 (0.86) CREB1ABCB1CYP3A4MAPTCYP2C9
SCHEMBL972407 0.90 CREB1 (1.00) CREB1ABCB1CYP3A4MAPTCYP2C9
SCHEMBL972837 0.87 CREB1 (0.80) CREB1ABCB1CYP3A4MAPTCYP2C9
SCHEMBL17663637 0.86 CREB1 (0.81) CREB1ABCB1CYP3A4MAPTCYP2C9
SCHEMBL972738 0.85 CREB1 (0.70) CREB1ABCB1CYP3A4MAPTCYP2C9
SCHEMBL22966700 0.84 ABCB1 (0.60) CREB1ABCB1CYP3A4MAPTCYP2C9
Baicalein SCHEMBL29200768 0.83 ABCB1 (0.89) CREB1ABCB1CYP3A4MAPTCYP2C9
SCHEMBL21224157 0.82 MAPT (0.74) CREB1ABCB1CYP3A4MAPTCYP2C9
SCHEMBL29494596 0.82 MAPT (0.74) CREB1ABCB1CYP3A4MAPTCYP2C9
SCHEMBL971180 0.82 CREB1 (0.66) CREB1ABCB1CYP3A4MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021026257-A1 PRODRUGS OF ALOX-15 INHIBITORS AND METHODS OF USING THE SAME EMPIRICO INC. (US) 2021-02-11 WO disclosed