SCHEMBL22978617

SCHEMBL22978617

CC1Cc2ccccc2OC1(C)N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MITF O75030 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
KDM1A O60341 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
PKM P14618 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
CYP2C19 P33261 1/20 0.33
THPO P40225 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
NISCH Q9Y2I1 1/20 0.33
MAOA P21397 8/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10382447 0.81 SMN1; SMN2 (0.36) SMN1; SMN2KDM4EMITFLMNAPOLB
SCHEMBL6723346 0.79 MAOA (0.36) SMN1; SMN2KDM4EMITFLMNAPOLB
SCHEMBL1820342 0.76 PTPN1 (0.36) SMN1; SMN2KDM4EMITFLMNAPOLB
SCHEMBL6171978 0.76 PARP1 (0.36) TSHRNISCHMAOB
SCHEMBL25273343 0.74 NPC1 (0.33) MAPK1
SCHEMBL10192535 0.74 MAOA (0.37) SMN1; SMN2KDM4EMITFLMNAPOLB
SCHEMBL28330440 0.73 TSHR (0.36) SMN1; SMN2KDM4EMITFLMNAPOLB
SCHEMBL787684 0.72 CREBBP (0.32) SMN1; SMN2KDM4EMITFLMNAPOLB
SCHEMBL16797653 0.71 CREBBP (0.36) SMN1; SMN2KDM4EMITFLMNAPOLB
SCHEMBL3310654 0.70 MGAM (0.47) KDM4EMAOAMAOBPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023102747-A1 ANTIMALARIAL AGENTS MERCK SHARP & DOHME LLC (US) 2023-06-15 WO disclosed
EP-4013742-A1 ANTIMALARIAL AGENTS Merck Sharp & Dohme Corp. (US) 2022-06-22 EP disclosed
WO-2021026884-A1 ANTIMALARIAL AGENTS MERCK SHARP & DOHME CORP. (US) 2021-02-18 WO disclosed
WO-2021027502-A1 ANTIMALARIAL AGENTS MERCK SHARP & DOHME CORP. (US) 2021-02-18 WO disclosed