SCHEMBL6171978

SCHEMBL6171978

CC1Cc2ccccc2OC1(C)C(N)=O

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.36
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
GABRA1 P14867 2/20 0.33
GABRB2 P47870 2/20 0.33
NISCH Q9Y2I1 1/20 0.33
NOTUM Q6P988 1/20 0.33
ATM Q13315 1/20 0.33
HSD11B1 P28845 2/20 0.32
GPBAR1 Q8TDU6 1/20 0.32
TP53 P04637 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15820173 0.82 DRD2 (0.36) HPGDTSHRGABRA1GABRB2NOTUM
SCHEMBL22978617 0.76 SMN1; SMN2 (0.34) TSHRNISCHMAOB
SCHEMBL6723346 0.76 MAOA (0.36) HPGDTSHRNISCHMAOB
SCHEMBL10382447 0.75 SMN1; SMN2 (0.36) TSHRNISCHMAOB
SCHEMBL27887531 0.73 ATM (0.42) ATM
SCHEMBL10192535 0.72 MAOA (0.37) NISCHMAOB
SCHEMBL1820342 0.70 PTPN1 (0.36) TSHRGABRA1GABRB2NISCHMAOB
SCHEMBL6650230 0.70 CYP3A4 (0.38) HPGDATM
SCHEMBL787684 0.70 CREBBP (0.32) PARP1
SCHEMBL8370012 0.68 MGAM (0.47) HPGDMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534693-A2 1, 3-DIAMINO-2-HYDROXYPROPANE PRODRUG DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2005-06-01 EP claimed
EP-1453789-A2 N,N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES Elan Pharmaceuticals, Inc. (US) 2004-09-08 EP claimed
WO-2004022523-A2 1, 3-DIAMINO-2-HYDROXYPROPANE PRODRUG DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2004-03-18 WO claimed
WO-2003040096-A2 N, N'-SUBSTITUTED-1,3-DIAMINO-2-HYDROXYPROPANE DERIVATIVES ELAN PHARMACEUTICALS, INC. (US) 2003-05-15 WO claimed