SCHEMBL22979308

SCHEMBL22979308

COc1ccc(-c2nc3c4cccc(S(C)(=O)=O)c4nc(N[C@@H]4CN(C(=O)O)CCNC4=O)n3n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
ADORA3 P0DMS8 10/20 0.38
MAPT P10636 4/20 0.37
THRB P10828 1/20 0.36
XDH P47989 1/20 0.36
ADORA2A P29274 3/20 0.35
ADORA1 P30542 2/20 0.35
ZAP70 P43403 1/20 0.34
SYK P43405 1/20 0.34
MAPK1 P28482 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
GAA P10253 1/20 0.34
HTT P42858 1/20 0.34
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979824 0.93 MAPT (0.38) ALDH1A1KDM4EPOLBADORA3MAPT
SCHEMBL29646350 0.90 MMP9 (0.40) ALDH1A1KDM4EPOLBADORA3MAPT
SCHEMBL22987685 0.90 MMP9 (0.40) ALDH1A1KDM4EPOLBADORA3MAPT
SCHEMBL22980168 0.89 KDM4E (0.40) ALDH1A1KDM4EPOLBADORA3MAPT
SCHEMBL22979352 0.87 BRD4 (0.32) ALDH1A1KDM4EADORA3ADORA2AADORA1
SCHEMBL22979411 0.87 KDM4E (0.41) ALDH1A1KDM4EPOLBADORA3MAPT
SCHEMBL22979362 0.86 MAPT (0.38) ALDH1A1KDM4EPOLBADORA3MAPT
SCHEMBL22979649 0.85 KDM4E (0.41) ALDH1A1KDM4EPOLBADORA3MAPT
SCHEMBL22979082 0.85 ADORA3 (0.37) ALDH1A1KDM4EPOLBADORA3MAPT
SCHEMBL22979873 0.85 ADORA3 (0.37) ALDH1A1KDM4EPOLBADORA3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4013508-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES Bayer Aktiengesellschaft (DE) 2022-06-22 EP disclosed
WO-2021028382-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES BAYER AKTIENGESELLSCHAFT (DE) 2021-02-18 WO disclosed