SCHEMBL22979512

SCHEMBL22979512

Cn1cc(-c2nc3c4cccc(Br)c4nc(N[C@@H]4CN(C(=O)O)CCNC4=O)n3n2)cn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 13/20 0.34
ADORA2A P29274 8/20 0.33
CREBBP Q92793 4/20 0.33
BRD4 O60885 2/20 0.33
ADORA1 P30542 9/20 0.33
ADORA2B P29275 4/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RPLP1 P05386 1/20 0.31
RPLP0 P05388 1/20 0.31
RPS17 P08708 1/20 0.31
RPSA P08865 1/20 0.31
RPS2 P15880 1/20 0.31
RPL35A P18077 1/20 0.31
RPL7 P18124 1/20 0.31
RPL17 P18621 1/20 0.31
RPS4Y1 P22090 1/20 0.31
RPS3 P23396 1/20 0.31
RPS12 P25398 1/20 0.31
RPL13 P26373 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22979734 0.91 CREBBP (0.35) ADORA3ADORA2ACREBBPBRD4ADORA1
SCHEMBL22979749 0.90 ADORA3 (0.32) ADORA3ADORA2AADORA1ADORA2BAURKA
SCHEMBL29645740 0.90 ADORA3 (0.32) ADORA3ADORA2AADORA1ADORA2BAURKA
SCHEMBL29649011 0.89 ADORA3 (0.35) ADORA3ADORA2AADORA1
SCHEMBL22988240 0.89 ADORA3 (0.35) ADORA3ADORA2AADORA1
SCHEMBL28730362 0.89 ADORA3 (0.35) ADORA3ADORA2AADORA1
SCHEMBL22979062 0.89 CREBBP (0.37) ADORA3ADORA2ACREBBPBRD4ADORA1
SCHEMBL22979352 0.89 BRD4 (0.32) ADORA3ADORA2ACREBBPBRD4ADORA1
SCHEMBL22979177 0.88 CREBBP (0.33) ADORA3ADORA2ACREBBPBRD4ADORA1
SCHEMBL22988306 0.87 ADORA2A (0.35) ADORA3ADORA2AADORA1ADORA2BRPLP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4013508-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES Bayer Aktiengesellschaft (DE) 2022-06-22 EP disclosed
WO-2021028382-A1 [1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES BAYER AKTIENGESELLSCHAFT (DE) 2021-02-18 WO disclosed