SCHEMBL22980195

SCHEMBL22980195

C#CC(CC(C)(C)C)OC(N)=O

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
MAPT P10636 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22980192 1.00 LMNA (0.33) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL29032631 0.81 LMNA (0.33) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL28635010 0.81 AOC1 (0.31)
SCHEMBL29032630 0.81 LMNA (0.33) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL5165702 0.73 CA2 (0.42) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL24372220 0.73 LMNA (0.39) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL29210106 0.71 LMNA (0.52) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL23629921 0.70 LMNA (0.32) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL31314516 0.69 LMNA (0.32) LMNACHRM2CHRM4CHRM5CHRM1
SCHEMBL16330481 0.69 LMNA (0.36) LMNACHRM2CHRM4CHRM5CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021115401-A1 FLUORINE-CONTAINING HETEROCYCLIC DERIVATIVES WITH MACROCYCLIC STRUCTURE AND USE THEREOF 成都倍特药业股份有限公司 2021-06-17 WO disclosed
WO-2021042890-A1 HETEROCYCLIC COMPOUND AND APPLICATION THEREOF AS TRK KINASE INHIBITOR 罗欣药业(上海)有限公司 2021-03-11 WO disclosed
WO-2021027503-A1 TRICYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND INTERMEDIATE AND USE THEREOF 罗欣药业(上海)有限公司 2021-02-18 WO disclosed