SCHEMBL22980312

SCHEMBL22980312

CN1C(=O)COc2c(Br)cccc21.O=C1COc2c(Br)cccc2N1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.40
DRD2 P14416 5/20 0.40
HTR1D P28221 5/20 0.39
HTR1B P28222 5/20 0.39
SLC6A4 P31645 5/20 0.39
KCNH2 Q12809 4/20 0.39
BRPF1 P55201 1/20 0.38
HTR2A P28223 1/20 0.38
PDE3B Q13370 3/20 0.37
PDE3A Q14432 3/20 0.37
KMT2A Q03164 1/20 0.37
SMYD3 Q9H7B4 1/20 0.36
TRPV1 Q8NER1 1/20 0.35
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16361881 0.87 HTR1A (0.41) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL29736794 0.84 SMYD3 (0.45) HTR1ADRD2HTR1DHTR1BSLC6A4
SCHEMBL2380905 0.84 SMYD3 (0.45) HTR1ADRD2HTR1DHTR1BSLC6A4
SCHEMBL3593642 0.72 HTR1A (0.41) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL2172798 0.71 PKM (0.44) KMT2ASMYD3BRD4CREBBP
SCHEMBL14867323 0.70 HTR1A (0.44) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL4484367 0.69 NPC1 (0.41) HTR1AKMT2ASMYD3BRD4CREBBP
SCHEMBL474683 0.69 TERT (0.47) HTR1AHTR1DHTR1BSLC6A4KCNH2
SCHEMBL1851941 0.69 CREBBP (0.58) HTR1ADRD2HTR1DHTR1BSLC6A4
SCHEMBL254031 0.69 SMYD3 (0.48) HTR1ADRD2KMT2ASMYD3BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4010335-A1 SHP2 INHIBITORS IRBM S.P.A. (IT) 2022-06-15 EP disclosed
WO-2021028362-A1 SHP2 INHIBITORS IRBM S.P.A. (IT) 2021-02-18 WO disclosed