SCHEMBL2298330

SCHEMBL2298330

CC/C(=C\C(=O)O)c1cc(C)c(Oc2ccc(OCc3cscn3)cn2)c(C)c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ALOX5 P09917 2/20 0.33
SCD O00767 1/20 0.33
PPARG P37231 1/20 0.31
PKM P14618 1/20 0.31
ALOX5AP P20292 1/20 0.31
ACACB O00763 2/20 0.30
ACACA Q13085 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2298336 0.84 ESR1 (0.36) MAPK14MAPK1NPSR1ALOX5SCD
SCHEMBL2231441 0.84 PDE10A (0.37) PPARGALOX5AP
SCHEMBL13582005 0.82 CYP4F2 (0.36) ALOX5PPARGPKM
SCHEMBL13582003 0.82 CYP4F2 (0.36) ALOX5PPARGPKM
SCHEMBL2232840 0.80 MAPT (0.35)
SCHEMBL2298327 0.78 CA12 (0.38)
SCHEMBL2231791 0.67 PPARG (0.40) ALOX5PPARGACACBACACA
SCHEMBL2235842 0.67 TDP1 (0.37) MAPK1ALOX5PPARG
SCHEMBL2231445 0.67 HTR2A (0.36) ALOX5PPARGALOX5AP
SCHEMBL2233200 0.67 ALOX5 (0.35) ALOX5PPARGALOX5APACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed