SCHEMBL2298336

SCHEMBL2298336

CCC(=Cc1cc(C)c(Oc2ccc(OCc3cscn3)cn2)c(C)c1)C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.36
ALOX5 P09917 4/20 0.35
CTSD P07339 1/20 0.32
BACE1 P56817 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
SCD O00767 1/20 0.32
MAPK14 Q16539 2/20 0.32
TBXAS1 P24557 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALOX5AP P20292 1/20 0.31
ACACB O00763 2/20 0.30
ACACA Q13085 2/20 0.30
PSEN1 P49768 1/20 0.30
PPARG P37231 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13582005 0.84 CYP4F2 (0.36) ESR1ALOX5KDM4EPPARG
SCHEMBL13582003 0.84 CYP4F2 (0.36) ESR1ALOX5KDM4EPPARG
SCHEMBL2231445 0.84 HTR2A (0.36) ESR1ALOX5ALOX5APPPARG
SCHEMBL2298330 0.84 MAPK14 (0.34) ALOX5MAPK1NPSR1SCDMAPK14
SCHEMBL2298327 0.82 CA12 (0.38) ESR1BACE1
SCHEMBL2232843 0.80 ESR1 (0.41) ESR1ALOX5TBXAS1KDM4EPSEN1
SCHEMBL2231793 0.67 PPARG (0.48) ALOX5PSEN1PPARG
SCHEMBL2235847 0.67 ALOX5 (0.41) ALOX5MAPK1PSEN1PPARG
SCHEMBL13582112 0.67 CYP4F2 (0.40) ESR1KDM4E
SCHEMBL13581834 0.67 RAB9A (0.43) ESR1KDM4EACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed