SCHEMBL2298746

SCHEMBL2298746

Fc1cc(Cl)ccc1OC1CNC1

nearest known ligand 0.72

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 10/20 0.58
HTR2C P28335 1/20 0.57
HTR2B P41595 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12374729 0.84 SLC6A4 (0.77) SLC6A4HTR2CHTR2B
SCHEMBL5367403 0.83 HTR2C (0.54) SLC6A4HTR2CHTR2B
SCHEMBL2298800 0.82 SLC6A4 (0.60) SLC6A4HTR2CHTR2B
SCHEMBL14956969 0.82 SLC6A4 (0.59) SLC6A4HTR2CHTR2B
SCHEMBL30945291 0.81 FPR2 (0.48) SLC6A4HTR2CHTR2B
Hydrochloric Acid SCHEMBL30357915 0.81 SLC6A4 (0.57) SLC6A4HTR2CHTR2B
SCHEMBL23255234 0.79 SLC6A4 (0.51) SLC6A4HTR2CHTR2B
SCHEMBL14957073 0.79 SLC6A4 (0.57) SLC6A4HTR2CHTR2B
SCHEMBL20425543 0.79 SLC6A4 (0.57) SLC6A4HTR2CHTR2B
SCHEMBL14054027 0.79 SLC6A2 (0.51) SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210292305-A1 Cyclic Ureas SIRONAX LTD (KY) 2021-09-23 US disclosed
US-9334269-B2 Carboxamides as inhibitors of voltage-gated sodium channels AMGEN INC. (US) 2016-05-10 US disclosed
US-20130131035-A1 CARBOXAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS AMGEN INC. (US) 2013-05-23 US disclosed
EP-2536689-A1 ARYL CARBOXAMIDE DERIVATIVES AS SODIUM CHANNEL INHIBITORS FOR TREATMENT OF PAIN Amgen Inc. (US) 2012-12-26 EP disclosed
WO-2011103196-A1 ARYL CARBOXAMIDE DERIVATIVES AS SODIUM CHANNEL INHIBITORS FOR TREATMENT OF PAIN AMGEN INC. (US) 2011-08-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130131035-A1 CARBOXAMIDES AS INHIBITORS OF VOLTAGE-GATED SODIUM CHANNELS CACNA1B, SCN1A, CACNA1I SLC6A4 502/4885HTR2C 379/4885HTR2B 373/4885
US-20210292305-A1 Cyclic Ureas RIPK1, RIPK3, RIPK4 SLC6A4 4608/4885HTR2C 3927/4885HTR2B 4192/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.