SCHEMBL2299273

SCHEMBL2299273

CC(C)c1cc(C(C)C)c(-c2cccc(C(C)(C)C)c2P)c(C(C)C)c1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.34
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
CA2 P00918 1/20 0.32
FABP3 P05413 2/20 0.31
FABP4 P15090 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
FABP5 Q01469 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30317598 0.85 ROCK2 (0.39) ROCK2GABRA1GABRB2CA2FABP3
Hydrochloric Acid SCHEMBL21331878 0.84 ROCK2 (0.38) ROCK2GABRA1GABRB2CA2FABP3
SCHEMBL29382588 0.83 ROCK2 (0.35) ROCK2GABRA1GABRB2CA2FABP3
SCHEMBL1728407 0.81 GABRA1 (0.31) GABRA1GABRB2FABP3FABP4CYP1A2
SCHEMBL3432179 0.78 ROCK2 (0.34) ROCK2
SCHEMBL366622 0.74 GABRA1 (0.37) ROCK2GABRA1GABRB2CA2FABP3
SCHEMBL14929520 0.72 ROCK2 (0.35) ROCK2GABRA1GABRB2CA2FABP3
SCHEMBL16050488 0.72 GABRA1 (0.52) ROCK2GABRA1GABRB2CA2FABP3
SCHEMBL16050486 0.72 FABP3 (0.41) ROCK2GABRA1GABRB2CA2FABP3
SCHEMBL3684193 0.72 GABRA1 (0.47) GABRA1GABRB2CA2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011103460-A1 FUSED TETRACYCLIC PYRIDO[4,3-B]INDOLE AND PYRIDO[3,4-B]ONDOLE DERIVATIVES AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2011-08-25 WO disclosed
WO-2011103433-A1 PYRIDO[4,3-B]INDOLE AND PYRIDO[3,4-B]INDOLE DERIVATIVES AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2011-08-25 WO disclosed