SCHEMBL2299449

SCHEMBL2299449

C=Cc1ccc(Br)cc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.42
HCAR1 Q9BXC0 1/20 0.39
NT5E P21589 1/20 0.39
APP P05067 1/20 0.36
NPFFR1 Q9GZQ6 1/20 0.35
NPFFR2 Q9Y5X5 1/20 0.35
SLC22A12 Q96S37 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
MTOR P42345 1/20 0.32
HTT P42858 1/20 0.32
NCOA1 Q15788 1/20 0.32
NCOA3 Q9Y6Q9 1/20 0.32
HRH4 Q9H3N8 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
CDK1 P06493 1/20 0.31
CDK4 P11802 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL207592 0.80 ERN1 (0.47) KDM1AHCAR1NT5EAPPALDH1A1
SCHEMBL1130682 0.78 IDO1 (0.42) HCAR1APP
SCHEMBL4076004 0.78 CES2 (0.46) HCAR1APPKDM4E
SCHEMBL3702783 0.76 APP (0.51) APPALDH1A1LMNAHTTMAOB
SCHEMBL21880623 0.76 SMN1; SMN2 (0.38) APPKDM4ELMNAHTTNCOA1
SCHEMBL9996387 0.76 HCAR1 (0.39) HCAR1APPKDM4EALDH1A1
SCHEMBL2790893 0.76 GAA (0.55) APPKDM4EALDH1A1HPGD
SCHEMBL30950877 0.76 GAA (0.55) APPKDM4EALDH1A1HPGD
SCHEMBL1436520 0.76 HPGD (0.44) KDM1AHCAR1NT5EAPPNPFFR1
SCHEMBL1436519 0.76 HPGD (0.44) KDM1AHCAR1NT5EAPPNPFFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109880065-B Conjugated polymer containing trifluoromethyl as well as preparation method and application thereof 中国科学院化学研究所 2020-05-26 CN disclosed
WO-2011103063-A1 THERAPEUTIC COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-08-25 WO disclosed