SCHEMBL207592

SCHEMBL207592

O=Cc1ccc(Br)cc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 4/20 0.47
HCAR1 Q9BXC0 1/20 0.42
KDM1A O60341 2/20 0.42
CYP2A6 P11509 2/20 0.41
NT5E P21589 1/20 0.39
PTPN1 P18031 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
ALDH1A1 P00352 1/20 0.36
KIF11 P52732 1/20 0.36
APP P05067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30217843 0.84 ERN1 (0.52) ERN1HCAR1KDM1ACYP2A6NT5E
SCHEMBL28949295 0.84 ERN1 (0.52) ERN1HCAR1KDM1ACYP2A6NT5E
SCHEMBL2299449 0.80 KDM1A (0.42) ERN1HCAR1KDM1ANT5EALDH1A1
SCHEMBL333114 0.78 IDO1 (0.42) ERN1HCAR1PTPN1ALDH1A1KIF11
SCHEMBL6852469 0.78 APP (0.49) ERN1ALDH1A1KIF11APP
SCHEMBL472401 0.78 CES2 (0.50) ERN1HCAR1KIF11APP
SCHEMBL10408709 0.76 ALDH1A1 (0.42) ERN1CYP2A6ALDH1A1KIF11APP
SCHEMBL1781235 0.76 ERN1 (0.52) ERN1KDM1ACYP2A6NT5EPTPN1
SCHEMBL502871 0.76 TDP1 (0.55) ERN1HCAR1PTPN1KIF11APP
SCHEMBL3718412 0.76 APP (0.51) ERN1ALDH1A1KIF11APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 134 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025224085-A1 COMPOUNDS CAPABLE OF ACTING ON S1R AS WELL AS ON SEH AND USES THEREOF UNIVERSITAT DE BARCELONA (ES) 2025-10-30 WO disclosed
US-20250304568-A1 PYRIMIDINES FOR DEGRADING BRUTON'S TYROSINE KINASE ABBVIE INC (US) 2025-10-02 US disclosed
US-20250122223-A1 HETEROCYCLIC COMPOUNDS AS UBIQUITIN SPECIFIC PROTEASE 7 INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2025-04-17 US disclosed
CN-116410756-B Liquid crystal compound containing polyfluorofenanthrene structure and application thereof 北京云基科技股份有限公司 2025-04-11 CN disclosed
US-12258340-B2 Pyrazole MAGL inhibitors H. LUNDBECK A/S (DK) 2025-03-25 US disclosed
CN-116473965-B Pyrazole MAGL inhibitors H.隆德贝克有限公司 2025-03-18 CN disclosed
US-20250026742-A1 COMPOUND AS ATR KINASE INHIBITOR SUZHOU ARK BIOPHARMACEUTICAL CO., LTD. (CN) 2025-01-23 US disclosed
EP-4480482-A2 PYRIMIDINES FOR DEGRADING BRUTON'S TYROSINE KINASE AbbVie Inc. (US) 2024-12-25 EP disclosed
US-12172992-B2 Pyrimidines for degrading Bruton's tyrosine kinase ABBVIE INC. (US) 2024-12-24 US disclosed
CN-115703768-B Compounds useful as inhibitors of ATR kinase 苏州爱科百发生物医药技术有限公司 2024-12-17 CN disclosed
CN-101541747-A Biphenyl amide lactam derivatives as inhibitors of 11- beta-hydroxysteroid dehydrogenase 1 LILLY CO ELI (US) 2009-09-23 CN disclosed
US-20090197880-A1 ANTI-VIRAL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE GENELABS TECHNOLOGIES, INC. 2009-08-06 US disclosed
US-20090156571-A1 BIPHENYL AMIDE LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY 2009-06-18 US disclosed
EP-2049481-A2 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SmithKline Beecham Corporation (US) 2009-04-22 EP disclosed
EP-2016047-A1 BIPHENYL AMIDE LACTAM DERIVATIVES AS INHIBITORS OF 11- BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2009-01-21 EP disclosed
US-20080261920-A1 2-Aminooxazolines as TAAR1 ligands F. HOFFMANN-LA ROCHE AG (CH) 2008-10-23 US disclosed
WO-2008092785-A1 NOVEL 2-AMINOOXAZOLINES AS TAAR1 LIGANDS FOR CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2008-08-07 WO disclosed
WO-2008021851-A2 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-21 WO disclosed
WO-2008021851-A2 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS FOR OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-21 WO disclosed
WO-2007124337-A1 BIPHENYL AMIDE LACTAM DERIVATIVES AS INHIBITORS OF 11- BETA-HYDROXYSTEROID DEHYDROGENASE 1 ELI LILLY AND COMPANY (US) 2007-11-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250304568-A1 PYRIMIDINES FOR DEGRADING BRUTON'S TYROSINE KINASE BTK, TYMP, LYN ERN1 223/4885HCAR1 2098/4885KDM1A 568/4885
US-20250026742-A1 COMPOUND AS ATR KINASE INHIBITOR ATR, CHEK2, CHEK1 ERN1 460/4885HCAR1 4570/4885KDM1A 1908/4885
US-12258340-B2 Pyrazole MAGL inhibitors MGLL, PNLIP, LPL ERN1 1174/4885HCAR1 3754/4885KDM1A 2496/4885
US-20250122223-A1 HETEROCYCLIC COMPOUNDS AS UBIQUITIN SPECIFIC PROTEASE 7 INHIBITORS USP7, UBA7, SENP7 ERN1 1151/4885HCAR1 3348/4885KDM1A 303/4885
US-20090197880-A1 ANTI-VIRAL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE HAVCR2, SARS1, RPL35 ERN1 487/4885HCAR1 4669/4885KDM1A 3691/4885
US-20090156571-A1 BIPHENYL AMIDE LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 HSD11B1, HSD17B1, HSD11B2 ERN1 1347/4885HCAR1 179/4885KDM1A 251/4885
US-20080261920-A1 2-Aminooxazolines as TAAR1 ligands TAAR1, TAAR5, NPY2R ERN1 3566/4885HCAR1 77/4885KDM1A 2377/4885
US-12172992-B2 Pyrimidines for degrading Bruton's tyrosine kinase BTK, TYMP, LYN ERN1 223/4885HCAR1 2098/4885KDM1A 568/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.