SCHEMBL2300600

SCHEMBL2300600

CN(c1ccc(NC(=O)c2ccc(N3CCNCC3)cc2)cn1)C1CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK7 Q13164 1/20 0.48
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
MCHR1 Q99705 7/20 0.46
NPC1 O15118 5/20 0.44
RAB9A P51151 5/20 0.44
MAPT P10636 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
MCL1 Q07820 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TP53 P04637 2/20 0.43
MAPK1 P28482 2/20 0.43
ALOX15 P16050 2/20 0.43
HTT P42858 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3345597 0.87 NPC1 (0.48) MAPK7MCHR1NPC1RAB9AMAPT
SCHEMBL2303204 0.82 SMN1; SMN2 (0.56) MAPTSMN1; SMN2KMT2AMEN1LMNA
SCHEMBL24891825 0.77 RAB9A (0.64) ITGB3ITGA2BNPC1RAB9AMAPT
SCHEMBL2300598 0.76 HRH4 (0.51) ITGB3ITGA2BNPC1RAB9AMAPT
SCHEMBL17607243 0.75 MAPK7 (0.47) MAPK7NPC1RAB9A
SCHEMBL17801122 0.74 NPC1 (0.75) ITGB3ITGA2BNPC1RAB9AMAPT
SCHEMBL1663115 0.73 ALDH1A1 (0.66) ITGB3ITGA2BNPC1RAB9AMAPT
SCHEMBL8769785 0.73 RAB9A (0.59) ITGB3ITGA2BNPC1RAB9AMAPT
SCHEMBL24891642 0.73 MAPT (0.61) ITGB3ITGA2BNPC1RAB9AMAPT
SCHEMBL30182512 0.73 MAPT (0.61) ITGB3ITGA2BNPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350311-A1 DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS Via Pharmaceuticals, Inc. (US) 2011-08-03 EP disclosed