SCHEMBL17607243

SCHEMBL17607243

CN(c1ccc(NC(=O)c2ccc[nH]2)cn1)C1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK7 Q13164 1/20 0.47
KDM1A O60341 1/20 0.42
RCOR1 Q9UKL0 1/20 0.42
SCN9A Q15858 1/20 0.42
TMIGD3 P0DMS9 1/20 0.42
ADORA1 P30542 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
GFER P55789 1/20 0.41
TRPV1 Q8NER1 1/20 0.38
S1PR1 P21453 4/20 0.38
S1PR3 Q99500 1/20 0.36
PIK3CA P42336 2/20 0.36
MTOR P42345 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17607239 0.76 TMIGD3 (0.46) MAPK7KDM1ARCOR1SCN9ATMIGD3
SCHEMBL20265732 0.75 MAPK7 (0.82) MAPK7
SCHEMBL2300600 0.75 MAPK7 (0.48) MAPK7NPC1RAB9A
SCHEMBL4072949 0.73 S1PR1 (0.49) MAPK7TRPV1S1PR1S1PR3PIK3CA
SCHEMBL17607174 0.72 MAPK7 (0.58) MAPK7KDM1ARCOR1SCN9ATMIGD3
SCHEMBL4068903 0.70 NPC1 (0.51) NPC1RAB9ATRPV1S1PR1PIK3CA
SCHEMBL4063941 0.70 S1PR1 (0.51) MAPK7NPC1RAB9ATRPV1S1PR1
SCHEMBL4069506 0.69 SMN1; SMN2 (0.54) MAPK7NPC1RAB9ATRPV1S1PR1
SCHEMBL3345597 0.68 NPC1 (0.48) MAPK7NPC1RAB9A
SCHEMBL5483909 0.67 SMN1; SMN2 (0.53) NPC1RAB9AGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3194390-A1 PYRROLCARBOXAMIDE DERIVATIVES FOR THE INHBITION OF ERK5 Cancer Research Technology Ltd (GB) 2017-07-26 EP claimed
WO-2016042341-A1 PYRROLCARBOXAMIDE DERIVATIVES FOR THE INHBITION OF ERK5 CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2016-03-24 WO claimed