SCHEMBL2301357

SCHEMBL2301357

CCCCCCCC/C=C\CCCCCCCCOC(C)(CN(C)C)OCCCCCCCC/C=C\CCCCCCCC

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LPAR2 Q9HBW0 3/20 0.44
LPAR3 Q9UBY5 3/20 0.44
LPAR1 Q92633 2/20 0.44
FAAH O00519 2/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12462210 0.95 ALDH1A1 (0.45)
SCHEMBL14715889 0.95 ALDH1A1 (0.45)
SCHEMBL6263292 0.91 DNM1 (0.39)
SCHEMBL2519902 0.91 DNM1 (0.39)
SCHEMBL935452 0.90 ALDH1A1 (0.41)
Trimethylammonium SCHEMBL3917836 0.81 LPAR2 (0.42) LPAR2LPAR3LPAR1FAAHTRPV1
SCHEMBL18184028 0.80 LPAR2 (0.50) LPAR2LPAR3LPAR1FAAHTRPV1
SCHEMBL16311960 0.80 LPAR2 (0.50) LPAR2LPAR3LPAR1FAAHTRPV1
SCHEMBL28438320 0.79 CNR1 (0.42) LPAR2LPAR3LPAR1FAAHTRPV1
SCHEMBL6831358 0.76 LPAR2 (0.44) LPAR2LPAR3LPAR1FAAHTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024119074-A1 STEALTH LIPID NANOPARTICLE COMPOSITIONS FOR CELL TARGETING GENERATION BIO CO. (US) 2024-06-06 WO claimed
CN-118043068-A RNA vaccine 阿克丘勒斯治疗公司 2024-05-14 CN claimed
WO-2019161263-A1 LIPID-SURFACTANT NANOPARTICLES FOR DRUG DELIVERY AND METHODS OF MAKING AND USES THEREOF OHIO STATE INNOVATION FOUNDATION (US) 2019-08-22 WO claimed
EP-3247328-A1 METHODS, COMPOSITIONS, AND SYSTEMS FOR DELIVERING THERAPEUTIC AND DIAGNOSTIC AGENTS INTO CELLS PhaseRx, Inc. (US) 2017-11-29 EP claimed
WO-2016118697-A9 METHODS, COMPOSITIONS, AND SYSTEMS FOR DELIVERING THERAPEUTIC AND DIAGNOSTIC AGENTS INTO CELLS PHASERX, INC. (US) 2016-09-29 WO claimed
WO-2016118697-A1 METHODS, COMPOSITIONS, AND SYSTEMS FOR DELIVERING THERAPEUTIC AND DIAGNOSTIC AGENTS INTO CELLS PHASERX, INC. (US) 2016-07-28 WO claimed
EP-4370135-A2 SINGLE CHAIN VARIABLE FRAGMENT (SCFV) MODIFIED LIPID NANOPARTICLE COMPOSITIONS AND USES THEREOF Generation Bio Co. (US) 2024-05-22 EP disclosed
CN-118043068-A RNA vaccine 阿克丘勒斯治疗公司 2024-05-14 CN disclosed
EP-4181948-A2 METHODS FOR ENCAPSULATING POLYNUCLEOTIDES INTO REDUCED SIZES OF LIPID NANOPARTICLES AND NOVEL FORMULATION THEREOF Generation Bio Co. (US) 2023-05-24 EP disclosed
WO-2023069628-A2 COMPOSITIONS AND METHODS FOR SILENCING KRAS NANOTHERA BIOSCIENCES, INC. (US) 2023-04-27 WO disclosed
WO-2023287861-A2 SINGLE CHAIN VARIABLE FRAGMENT (SCFV) MODIFIED LIPID NANOPARTICLE COMPOSITIONS AND USES THEREOF GENERATION BIO CO. (US) 2023-01-19 WO disclosed
WO-2022016089-A2 METHODS FOR ENCAPSULATING POLYNUCLEOTIDES INTO REDUCED SIZES OF LIPID NANOPARTICLES AND NOVEL FORMULATION THEREOF GENERATION BIO CO. (US) 2022-01-20 WO disclosed
EP-3934700-A1 NON-ACTIVE LIPID NANOPARTICLES WITH NON-VIRAL, CAPSID FREE DNA Generation Bio Co. (US) 2022-01-12 EP disclosed
EP-3247328-A1 METHODS, COMPOSITIONS, AND SYSTEMS FOR DELIVERING THERAPEUTIC AND DIAGNOSTIC AGENTS INTO CELLS PhaseRx, Inc. (US) 2017-11-29 EP disclosed
WO-2016118697-A9 METHODS, COMPOSITIONS, AND SYSTEMS FOR DELIVERING THERAPEUTIC AND DIAGNOSTIC AGENTS INTO CELLS PHASERX, INC. (US) 2016-09-29 WO disclosed
WO-2016118697-A1 METHODS, COMPOSITIONS, AND SYSTEMS FOR DELIVERING THERAPEUTIC AND DIAGNOSTIC AGENTS INTO CELLS PHASERX, INC. (US) 2016-07-28 WO disclosed
EP-2350043-A1 IMPROVED AMINO LIPIDS AND METHODS FOR THE DELIVERY OF NUCLEIC ACIDS TEKMIRA Pharmaceuticals Corporation (CA) 2011-08-03 EP disclosed
EP-2224912-A1 IMPROVED COMPOSITIONS AND METHODS FOR THE DELIVERY OF NUCLEIC ACIDS TEKMIRA Pharmaceuticals Corporation (CA) 2010-09-08 EP disclosed
WO-2010042877-A1 IMPROVED AMINO LIPIDS AND METHODS FOR THE DELIVERY OF NUCLEIC ACIDS TEKMIRA PHARMACEUTICALS CORPORATION (CA) 2010-04-15 WO disclosed
WO-2009086558-A1 IMPROVED COMPOSITIONS AND METHODS FOR THE DELIVERY OF NUCLEIC ACIDS TEKMIRA PHARMACEUTICALS CORPORATION (CA) 2009-07-09 WO disclosed