SCHEMBL2301756

SCHEMBL2301756

O=C(O)c1ccc(OC(=O)C2Nc3ccccc3C23CCNC3)cc1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ELANE P08246 3/20 0.36
ACHE P22303 4/20 0.35
BCHE P06276 2/20 0.35
SRD5A2 P31213 3/20 0.35
PKM P14618 1/20 0.35
POLB P06746 1/20 0.34
HSD17B10 Q99714 1/20 0.34
BACE1 P56817 1/20 0.34
MAPT P10636 1/20 0.33
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
KDM1A O60341 1/20 0.32
ALDH1A1 P00352 1/20 0.32
OPRD1 P41143 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2302824 0.89 KMT2A (0.40) ACHEBCHEPOLBMAPTALDH1A1
SCHEMBL14311949 0.81 BACE1 (0.43) ACHEBCHEBACE1MAPTKDM1A
SCHEMBL28998851 0.68 BACE1 (0.43) BACE1KDM1A
SCHEMBL6219295 0.65 L3MBTL1 (0.40) POLB
SCHEMBL8839080 0.63 RXRA (0.61) ELANEHSD17B10RXRARXRBRXRG
SCHEMBL24736421 0.62 HTR2A (0.42) HSD17B10BACE1KDM1AALDH1A1
SCHEMBL11672849 0.61 SRD5A2 (0.62) ELANESRD5A2PKMHSD17B10
SCHEMBL12891019 0.60 KDM1A (0.46) BACE1KDM1AALDH1A1
SCHEMBL28453797 0.60 KDM1A (0.36) POLBBACE1KDM1AALDH1A1
SCHEMBL1756160 0.60 KMT2A (0.54) ELANESRD5A2POLBHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536731-A1 SUBSTITUTED SPIROINDOLINONES F. Hoffmann-La Roche AG (CH) 2012-12-26 EP claimed
WO-2011101297-A1 SUBSTITUTED SPIROINDOLINONES F. HOFFMANN-LA ROCHE AG (CH) 2011-08-25 WO claimed