SCHEMBL2301904

SCHEMBL2301904

FC(F)(F)Oc1cc(I)cc(Cl)n1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 1/20 0.32
PGK1 P00558 1/20 0.30
KCNN3 Q9UGI6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2528479 0.81
SCHEMBL2301663 0.77 PGK1 (0.33) PGK1KCNN3
SCHEMBL11955179 0.77 PGK1 (0.33) PGK1KCNN3
SCHEMBL7807011 0.76 ATF1 (0.34) IGF1RPGK1KCNN3
SCHEMBL9586268 0.74 IGF1R (0.32) IGF1RPGK1KCNN3
SCHEMBL13172417 0.74 TRPV1 (0.34) PGK1KCNN3
SCHEMBL18398967 0.74 SMN1; SMN2 (0.36)
SCHEMBL7808650 0.73 KMT2A (0.50)
SCHEMBL13194452 0.73 KCNN3 (0.39) PGK1KCNN3
SCHEMBL16635330 0.73 LOXL2 (0.38) PGK1KCNN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210300943-A1 OGA INHIBITOR COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2021-09-30 US disclosed
EP-3810593-A1 OGA INHIBITOR COMPOUNDS Janssen Pharmaceutica NV (BE) 2021-04-28 EP disclosed
EP-3810136-A1 OGA INHIBITOR COMPOUNDS Janssen Pharmaceutica NV (BE) 2021-04-28 EP disclosed
US-20210115040-A1 OGA INHIBITOR COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2021-04-22 US disclosed
CN-112334461-A OGA inhibitor compounds 詹森药业有限公司 2021-02-05 CN disclosed
CN-112312908-A OGA inhibitor compounds 詹森药业有限公司 2021-02-02 CN disclosed
WO-2019243528-A1 OGA INHIBITOR COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2019-12-26 WO disclosed
WO-2019243526-A1 OGA INHIBITOR COMPOUNDS JANSSEN PHARMACEUTICA NV (BE) 2019-12-26 WO disclosed
EP-2350008-B1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES BAYER CROPSCIENCE AG (DE) 2012-09-05 EP disclosed
EP-2350008-A1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES Bayer CropScience AG (DE) 2011-08-03 EP disclosed
WO-2010040461-A1 METHOD FOR THE PREPARATION OF FUNCTIONALIZED TRIHALOMETHOXY SUBSTITUTED PYRIDINES BAYER CROPSCIENCE AG (DE) 2010-04-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210300943-A1 OGA INHIBITOR COMPOUNDS OGA, OGT, GRN IGF1R 2318/4885PGK1 193/4885KCNN3 4050/4885
US-20210115040-A1 OGA INHIBITOR COMPOUNDS OGA, OGT, GRN IGF1R 2318/4885PGK1 193/4885KCNN3 4050/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.