SCHEMBL23019331

SCHEMBL23019331

Nc1ncc(Cl)c(N2CCOCC2)n1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 13/20 0.49
MTOR P42345 6/20 0.49
PIK3R1 P27986 4/20 0.49
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
MAPT P10636 1/20 0.47
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
HRH4 Q9H3N8 1/20 0.45
NOS1 P29475 1/20 0.45
DHFR P00374 1/20 0.45
RICTOR Q6R327 1/20 0.45
RPTOR Q8N122 1/20 0.45
MAPKAP1 Q9BPZ7 1/20 0.45
MLST8 Q9BVC4 1/20 0.45
PIK3CD O00329 3/20 0.44
PIK3CB P42338 2/20 0.44
NUDT1 P36639 1/20 0.44
PIK3CG P48736 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1935491 0.83 KDM4E (0.46) CYP1A2CYP2D6MAPTKDM4EGAA
SCHEMBL18072393 0.80 PIK3CA (0.54) PIK3CAMTORPIK3R1KDM4EGAA
SCHEMBL14541937 0.80 KDM4E (0.69) PIK3CAMTORPIK3R1MAPTKDM4E
SCHEMBL7712459 0.80 ALDH1A1 (0.63) PIK3CAMTORPIK3R1KDM4EGAA
SCHEMBL3721187 0.78 PIK3CD (0.56) PIK3CAMTORPIK3R1MAPTGAA
SCHEMBL7714561 0.78 KDM4E (0.56) PIK3CAMTORPIK3R1KDM4EGAA
SCHEMBL7282145 0.78 CNR2 (0.56) PIK3CADHFR
SCHEMBL17059203 0.78 ALDH1A1 (0.46) MAPTKDM4E
SCHEMBL13650825 0.77 MAPT (0.54) PIK3CAMTORPIK3R1CYP1A2CYP2D6
SCHEMBL25598894 0.76 IKBKB (0.56) PIK3CAMTORPIK3R1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2021-02-24 EP disclosed