SCHEMBL7282145

SCHEMBL7282145

Nc1ncc(-c2cccc(Cl)c2Cl)c(N2CCOCC2)n1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 10/20 0.56
PTPN11 Q06124 3/20 0.47
DHFR P00374 1/20 0.47
PIK3CA P42336 2/20 0.46
LRRK2 Q5S007 1/20 0.46
CNR1 P21554 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272936 0.87 CNR2 (0.52) CNR2PTPN11CNR1
SCHEMBL7278447 0.85 PTPN11 (0.59) PTPN11
SCHEMBL3756924 0.78 NOS1 (0.66) CNR2PTPN11PIK3CA
SCHEMBL7714561 0.78 KDM4E (0.56) DHFRPIK3CA
SCHEMBL23019331 0.78 PIK3CA (0.49) DHFRPIK3CA
SCHEMBL7708544 0.78 NOS1 (0.58) DHFRPIK3CALRRK2
SCHEMBL6049559 0.73 FGFR1 (0.49) PTPN11DHFR
SCHEMBL975784 0.73 CYP2D6 (0.57) PTPN11DHFR
SCHEMBL7712374 0.73 PIK3CA (0.48) DHFRPIK3CA
SCHEMBL7712422 0.73 STK4 (0.54) DHFRPIK3CALRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0679645-A1 Pharmacologically active CNS pyridmidin compounds THE WELLCOME FOUNDATION LIMITED (GB) 1995-11-02 EP disclosed
EP-0459819-A2 Pharmacologically active CNS compound THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed