SCHEMBL23022293

SCHEMBL23022293

Cc1ccnc2c1CCN(C)C2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.35
HTR2B P41595 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP2C19 P33261 3/20 0.34
IKBKB O14920 1/20 0.34
RAF1 P04049 1/20 0.34
RPS6KB1 P23443 1/20 0.34
MAPK1 P28482 1/20 0.34
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
KDR P35968 1/20 0.34
MAPKAPK2 P49137 1/20 0.34
PRKAG1 P54619 1/20 0.34
MAP2K1 Q02750 1/20 0.34
PRKAA1 Q13131 1/20 0.34
NEK1 Q96PY6 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL403401 0.86 CYP2C19 (0.41) MAOAMAOBHTR2AHTR2CHTR2B
SCHEMBL17624447 0.85 CCR1 (0.35) HTR2AHTR2CHTR2BIKBKBRAF1
SCHEMBL256752 0.74 HTR2A (0.47) HTR2AHTR2CHTR2BKDM4E
SCHEMBL15290670 0.73 CYP2C19 (0.35) MAOAMAOBKDM4ECYP2C19ADRA2A
SCHEMBL795349 0.72 NOS3 (0.44) HTR2AHTR2CHTR2BKDM4EGRIN1
SCHEMBL795850 0.72 GRM4 (0.40) HTR2AHTR2CHTR2BKDM4EDRD1
SCHEMBL8271971 0.72 MAOA (0.40) MAOAMAOBHTR2CCYP2C19DRD2
SCHEMBL22993421 0.72 ALDH1A1 (0.36) MAOAMAOBHTR2AHTR2CHTR2B
SCHEMBL14295646 0.72 C5AR1 (0.46) KDM4EDRD2DRD4DRD3
SCHEMBL23198626 0.71 CHRM4 (0.41) MAOAMAOBKDM4ECYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021032148-A1 AMINOPYRAZINE COMPOUNDS AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2021-02-25 WO disclosed