Pentobarbital

Pentobarbital

SCHEMBL23045802

CCCC(C)C1(CC)C(=O)N=C([O-])NC1=O.[AlH3].[Na+]

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQ

The experimentally established mechanism targets of Pentobarbital. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GABRB3 known ✓ P28472 1/20 0.55
GABRA2 known ✓ P47869 1/20 0.55
GABRB2 known ✓ P47870 1/20 0.55
CYP3A4 P08684 3/20 0.55
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
OPRD1 P41143 1/20 0.55
LMNA P02545 3/20 0.53
MMP9 P14780 1/20 0.42
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
NR1I2 O75469 1/20 0.39
RECQL P46063 1/20 0.38
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pentobarbital SCHEMBL7033991 0.98 CYP3A4 (0.57) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL9221628 0.98 CYP3A4 (0.57) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL1247 0.98 CYP3A4 (0.57) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL2475274 0.97 CYP3A4 (0.55) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL21634384 0.97 CYP3A4 (0.55) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL11127769 0.97 CYP3A4 (0.55) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL11559632 0.97 CYP3A4 (0.55) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL9216527 0.97 CYP3A4 (0.55) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL6594849 0.97 CYP3A4 (0.55) CYP3A4KDM4EALDH1A1GABRB3OPRD1
Pentobarbital SCHEMBL1052470 0.97 CYP3A4 (0.55) CYP3A4KDM4EALDH1A1GABRB3OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024090867-A1 POLYETHYLENE RESIN HAVING EXCELLENT THERMAL RESISTANCE 주식회사 엘지화학 2024-05-02 WO disclosed
WO-2024090868-A1 POLYETHYLENE RESIN HAVING EXCELLENT HEAT RESISTANCE 주식회사 엘지화학 2024-05-02 WO disclosed
WO-2023172009-A1 ETHYLENE/1-HEXENE COPOLYMER HAVING IMPROVED LONG-TERM PHYSICAL PROPERTY STABILITY AND PROCESSABILITY 주식회사 엘지화학 2023-09-14 WO disclosed
WO-2023075115-A1 POLYETHYLENE RESIN COMPOSITION AND FILM COMPRISING SAME 주식회사 엘지화학 2023-05-04 WO disclosed
WO-2022071744-A1 ETHYLENE/1-HEXENE COPOLYMER HAVING EXCELLENT CONSTRUCTABILITY AND PROCESSABILITY 주식회사 엘지화학 2022-04-07 WO disclosed
WO-2021112623-A1 POLYPROPYLENE RESIN, POLYPROPYLENE FIBER AND METHOD FOR PREPARING SAME 주식회사 엘지화학 2021-06-10 WO disclosed
WO-2021083309-A1 METALLOCENE COMPOUND, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 中国石油化工股份有限公司 2021-05-06 WO disclosed
WO-2021071154-A1 POLYETHYLENE AND PREPARATION METHOD THEREFOR 주식회사 엘지화학 2021-04-15 WO disclosed
WO-2021066437-A1 ETHYLENE/1-HEXENE COPOLYMER HAVING EXCELLENT LONG-TERM PROPERTIES AND PROCESSIBILITY 주식회사 엘지화학 2021-04-08 WO disclosed
WO-2021066398-A1 PELLET-TYPE POLYPROPYLENE RESIN COMPOSITION AND PREPARATION METHOD THEREFOR 주식회사 엘지화학 2021-04-08 WO disclosed
WO-2021060907-A1 POLYETHYLENE, AND CHLORINATED POLYETHYLENE THEREOF 주식회사 엘지화학 2021-04-01 WO disclosed
WO-2021060908-A1 SUPPORTED HYBRID CATALYST AND METHOD FOR PREPARING POLYOLEFIN BY USING SAME 주식회사 엘지화학 2021-04-01 WO disclosed
WO-2021040425-A1 POLYPROPYLENE-BASED COMPOSITE AND METHOD FOR PRODUCING SAME 주식회사 엘지화학 2021-03-04 WO disclosed
WO-2021040139-A1 OLEFINIC COPOLYMER AND PREPARATION METHOD THEREFOR 주식회사 엘지화학 2021-03-04 WO disclosed