SCHEMBL23049705

SCHEMBL23049705

CCOC(=O)c1cc2cc(Cl)c(Br)cc2[nH]1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.63
KDM4E B2RXH2 3/20 0.60
ALDH1A1 P00352 3/20 0.60
HPGD P15428 3/20 0.60
RAB9A P51151 3/20 0.60
LMNA P02545 3/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
NPC1 O15118 2/20 0.60
MAPT P10636 2/20 0.60
KMT2A Q03164 2/20 0.60
MEN1 O00255 1/20 0.60
GLA P06280 1/20 0.60
GAA P10253 1/20 0.60
ATM Q13315 1/20 0.60
HSD17B10 Q99714 1/20 0.58
L3MBTL1 Q9Y468 2/20 0.54
HTT P42858 1/20 0.54
HRH3 Q9Y5N1 1/20 0.54
MMP13 P45452 8/20 0.53
MMP2 P08253 6/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22760538 0.94 ALOX15 (0.63) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL832201 0.88 ALOX15 (0.69) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL18331899 0.84 ALOX15 (0.64) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL1397950 0.84 KDM4E (0.62) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL18331701 0.83 ALOX15 (0.63) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL4395738 0.83 ALOX15 (0.63) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL30995155 0.83 KDM4E (0.60) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL30995161 0.83 KDM4E (0.60) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL4049040 0.83 ALOX15 (0.66) ALOX15KDM4EALDH1A1HPGDRAB9A
SCHEMBL1397951 0.82 ALDH1A1 (0.60) ALOX15KDM4EALDH1A1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3647311-B1 RHO-ASSOCIATED PROTEIN KINASE INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD AND USE THEREOF BEIJING TIDE PHARMACEUTICAL CO LTD (CN) 2023-11-01 EP disclosed
EP-3596064-B1 TOSYLACETATE BASED COMPOUNDS AND DERIVATIVES THEREOF AS PHGDH INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2021-03-03 EP disclosed