SCHEMBL23055267

SCHEMBL23055267

CC(C)Nc1ccn2cncc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.39
TBXAS1 P24557 1/20 0.38
NAMPT P43490 1/20 0.36
NTRK1 P04629 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
NR3C1 P04150 1/20 0.33
AXL P30530 1/20 0.32
BRD4 O60885 1/20 0.32
CREBBP Q92793 1/20 0.32
FASN P49327 1/20 0.31
PIM1 P11309 2/20 0.31
PIM2 Q9P1W9 2/20 0.31
CSNK2A1 P68400 1/20 0.31
PIM3 Q86V86 1/20 0.31
IDO1 P14902 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31
THRB P10828 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21646466 0.81 PRKCI (0.41) PRKCITBXAS1NAMPTNTRK1NR3C1
SCHEMBL25124500 0.77 TBXAS1 (0.40) PRKCITBXAS1NAMPTNTRK1NR3C1
SCHEMBL23432572 0.76 TBXAS1 (0.37) TBXAS1NAMPTTDP1NR3C1AXL
SCHEMBL17561679 0.74 TBXAS1 (0.40) PRKCITBXAS1NAMPTNTRK1NR3C1
SCHEMBL23055240 0.70 TDP1 (0.34) TDP1AXLALDH1A1LMNACYP3A4
SCHEMBL21037102 0.70 TBXAS1 (0.50) PRKCITBXAS1NAMPTNTRK1TDP1
SCHEMBL23055261 0.70 MAPK1 (0.36) TDP1ALDH1A1LMNACYP3A4THRB
SCHEMBL24629446 0.69 TBXAS1 (0.43) PRKCITBXAS1NAMPTNTRK1NR3C1
SCHEMBL23055242 0.68 PIK3CD (0.38) NAMPTNTRK1TDP1ALDH1A1LMNA
SCHEMBL23055259 0.68 IRAK4 (0.43) NAMPTNTRK1TDP1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021149767-A1 HETEROCYCLIC DERIVATIVE 大日本住友製薬株式会社 2021-07-29 WO disclosed
WO-2021039961-A1 RING-FUSED PYRAZOLE DERIVATIVE 大日本住友製薬株式会社 2021-03-04 WO disclosed