SCHEMBL2305656

SCHEMBL2305656

CC(=O)C(c1ccc(Cl)cc1)c1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.55
S1PR3 Q99500 1/20 0.55
ALDH1A1 P00352 1/20 0.54
CYP1A2 P05177 1/20 0.54
LMNA P02545 3/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
SLC6A3 Q01959 4/20 0.49
CHRM2 P08172 3/20 0.49
ADRA2B P18089 3/20 0.49
SLC6A2 P23975 3/20 0.49
SLC6A4 P31645 3/20 0.49
HRH1 P35367 3/20 0.49
KCNH2 Q12809 3/20 0.49
HRH3 Q9Y5N1 3/20 0.49
CHRM5 P08912 2/20 0.49
CHRM1 P11229 2/20 0.49
HRH2 P25021 2/20 0.49
HTR2A P28223 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14060543 0.87 ALDH1A1 (0.69) S1PR3ALDH1A1CYP1A2LMNANPSR1
SCHEMBL17858363 0.86 S1PR1 (0.56) S1PR1S1PR3ALDH1A1CYP1A2LMNA
SCHEMBL28144224 0.84 ALDH1A1 (0.54) S1PR1S1PR3ALDH1A1CYP1A2LMNA
SCHEMBL28251775 0.82 TSHR (0.56) ALDH1A1CYP1A2LMNANPSR1SLC6A3
SCHEMBL11822715 0.78 S1PR1 (0.48) S1PR1S1PR3ALDH1A1CYP1A2LMNA
SCHEMBL4441209 0.78 L3MBTL1 (0.51) S1PR1S1PR3ALDH1A1CYP1A2NPSR1
SCHEMBL28419252 0.78 BRD4 (0.55) S1PR1S1PR3SLC6A3CHRM2SLC6A2
SCHEMBL10882007 0.77 BRD4 (0.63) S1PR1S1PR3CYP1A2LMNABLM
SCHEMBL15470472 0.75 CHRM2 (0.55) S1PR1S1PR3ALDH1A1LMNABLM
SCHEMBL21246926 0.75 SLC6A2 (0.51) S1PR1S1PR3ALDH1A1LMNABLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349999-A1 ALLOSTERIC PROTEIN KINASE MODULATORS Universität des Saarlandes (DE) 2011-08-03 EP disclosed
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO disclosed