SCHEMBL23065087

SCHEMBL23065087

O=c1c2c(Cl)cccc2nc(Nc2ccccc2Cl)n1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 17/20 0.47
PIK3R1 P27986 12/20 0.47
PIK3CA P42336 4/20 0.46
PIK3CB P42338 4/20 0.46
PIK3CG P48736 3/20 0.46
KMT2A Q03164 1/20 0.45
PDE4B Q07343 1/20 0.44
PDE7A Q13946 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23065111 0.88 PIK3CD (0.48) PIK3CDPIK3R1PIK3CAPIK3CBPIK3CG
SCHEMBL23065093 0.87 TP53 (0.50) PIK3CDPIK3R1PIK3CAPIK3CBPIK3CG
SCHEMBL24089980 0.87 ALDH1A1 (0.51) KMT2APDE4BPDE7A
SCHEMBL23064692 0.81 TP53 (0.47)
SCHEMBL24089999 0.80 MAPT (0.50) KMT2APDE4BPDE7A
SCHEMBL23065144 0.80 PDE7A (0.52) PIK3CDPIK3CGPDE4BPDE7A
SCHEMBL24090125 0.79 PIK3CD (0.50) PIK3CDPIK3R1PIK3CAPIK3CBPIK3CG
SCHEMBL23065090 0.78 C1R (0.48) PDE4BPDE7A
SCHEMBL18923546 0.77 HRH3 (0.57) PIK3CDPIK3R1
SCHEMBL23065109 0.76 SMN1; SMN2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11352366-B2 2-aminoquinazolinone derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-06-07 US disclosed
US-20220143020-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-05-12 US disclosed
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-09 US disclosed
WO-2021039968-A1 2-AMINOQUINAZOLINONE DERIVATIVE 大日本住友製薬株式会社 2021-03-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220143020-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, CRKL PIK3CD 4554/4885PIK3R1 3904/4885PIK3CA 4389/4885
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, SLC26A3 PIK3CD 4497/4885PIK3R1 4054/4885PIK3CA 4289/4885
US-11352366-B2 2-aminoquinazolinone derivative CNKSR1, HAX1, SLC26A3 PIK3CD 4497/4885PIK3R1 4054/4885PIK3CA 4289/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.