Bicarbonate

Bicarbonate

SCHEMBL2306960

O=C(O)O.O=C(c1ccc(-c2ccc(Nc3nc4cc(F)c(F)cc4[nH]3)cc2)cc1)C1CCCC1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B known ✓ P49841 1/20 0.43
HDAC11 Q96DB2 1/20 0.49
CHEK2 O96017 2/20 0.46
POLB P06746 2/20 0.45
CSNK1A1 P48729 2/20 0.43
CSNK1D P48730 2/20 0.43
CSNK1G2 P78368 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
PIK3CA P42336 8/20 0.42
CSF1R P07333 1/20 0.42
MTOR P42345 7/20 0.41
HDAC6 Q9UBN7 1/20 0.41
PIK3CD O00329 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12430197 0.98 HDAC11 (0.51) HDAC11CHEK2POLBCSNK1A1CSNK1D
SCHEMBL12266215 0.90 HDAC11 (0.46) HDAC11CHEK2POLBCSNK1A1CSNK1D
SCHEMBL1748082 0.86 DGAT1 (0.50) HDAC11POLBDGAT1
SCHEMBL1748083 0.86 DGAT1 (0.50) HDAC11POLBDGAT1
SCHEMBL1748084 0.86 DGAT1 (0.50) HDAC11POLBDGAT1
Bicarbonate SCHEMBL2307781 0.84 P2RY14 (0.42) CHEK2POLBCSNK1A1CSNK1DCSNK1G2
Bicarbonate SCHEMBL2316045 0.84 SMN1; SMN2 (0.56) CHEK2POLBCSNK1A1CSNK1DCSNK1G2
Bicarbonate SCHEMBL2313113 0.82 RAB9A (0.47) CHEK2POLBKDM4EMEN1LMNA
Bicarbonate SCHEMBL2310230 0.79 NPC1 (0.52) CHEK2POLBKDM4EMEN1MAPT
Bicarbonate SCHEMBL2312392 0.77 DGAT1 (0.41) CHEK2POLBCSNK1DCSNK1G2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP claimed