Bicarbonate

Bicarbonate

SCHEMBL2310230

O=C(O)O.O=C(c1ccc(-c2ccc(Nc3nc4ccccc4[nH]3)c(F)c2)cc1)C1CCCC1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.52
RAB9A P51151 7/20 0.52
SMN1; SMN2 Q16637 5/20 0.52
POLB P06746 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
CYP1A2 P05177 1/20 0.44
DGAT1 O75907 2/20 0.43
CHEK2 O96017 1/20 0.43
AKR1C3 P42330 1/20 0.43
KDM4E B2RXH2 1/20 0.42
TP53 P04637 1/20 0.42
PKM P14618 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CSF1R P07333 1/20 0.42
MAPT P10636 1/20 0.42
MEN1 O00255 1/20 0.41
CASP3 P42574 1/20 0.41
KMT2A Q03164 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1748153 0.87 DGAT1 (0.59) NPC1RAB9ASMN1; SMN2POLBTDP1
SCHEMBL5984327 0.87 DGAT1 (0.59) NPC1RAB9ASMN1; SMN2POLBTDP1
Bicarbonate SCHEMBL2312392 0.87 DGAT1 (0.41) NPC1RAB9ASMN1; SMN2POLBTDP1
Bicarbonate SCHEMBL2307118 0.86 DGAT1 (0.46) NPC1RAB9ASMN1; SMN2DGAT1CHEK2
Bicarbonate SCHEMBL2316045 0.85 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2POLBTDP1
SCHEMBL1748064 0.83 DGAT1 (0.48) NPC1RAB9ASMN1; SMN2POLBTDP1
SCHEMBL1748065 0.83 DGAT1 (0.41) NPC1RAB9ASMN1; SMN2POLBTDP1
Bicarbonate SCHEMBL2309476 0.79 DGAT1 (0.63) NPC1RAB9ASMN1; SMN2POLBCYP1A2
Bicarbonate SCHEMBL2306960 0.79 HDAC11 (0.49) NPC1RAB9ASMN1; SMN2POLBTDP1
Bicarbonate SCHEMBL2310705 0.77 DGAT1 (0.65) NPC1RAB9APOLBCYP1A2DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633722-B1 PREPARATION AND USE OF ARYL ALKYL ACID DERIVATIVES FOR THE TREATMENT OF OBESITY BAYER HEALTHCARE LLC (US) 2011-08-03 EP claimed