SCHEMBL23071306

SCHEMBL23071306

O=C(O)CCc1n[nH]c(=O)n(-c2ccc(F)cc2)c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
PTGS2 P35354 1/20 0.38
FFAR1 O14842 1/20 0.38
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
POLB P06746 1/20 0.36
PDE10A Q9Y233 1/20 0.36
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
ALOX15 P16050 1/20 0.36
APEX1 P27695 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
NR1H4 Q96RI1 1/20 0.34
NPC1 O15118 1/20 0.34
CSNK2A1 P68400 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14969183 0.76 KMT2A (0.46) ALDH1A1TSHRHTTKDM4ETDP1
SCHEMBL23565181 0.73 ALDH1A1 (0.42) ALDH1A1TSHRHTTPOLBKDM4E
SCHEMBL23071277 0.73 POLB (0.41) RXRARXRBRXRGPTGS2POLB
SCHEMBL14968994 0.69 NPC1 (0.51) ALDH1A1HTTPOLBKDM4ENPC1
SCHEMBL1133466 0.67 TDP1 (0.66) ALDH1A1TSHRHTTPOLBKDM4E
SCHEMBL8186274 0.67 ALDH1A1 (0.44) ALDH1A1TSHRHTTPOLBTDP1
SCHEMBL23071006 0.67 PLA2G4A (0.46) ALDH1A1RXRARXRBRXRGPTGS2
SCHEMBL6476570 0.67 AR (0.53) ALDH1A1POLBNPC1
SCHEMBL7094306 0.66 MAPK9 (0.53) ALDH1A1POLBKDM4ETDP1NPC1
SCHEMBL23070989 0.66 PLA2G4A (0.36) ALDH1A1RXRARXRBRXRGPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021043217-A1 COMPOUND HAVING AXL AND C-MET KINASE INHIBITORY ACTIVITY, PREPARATION THEREOF AND APPLICATION THEREOF 中国科学院上海药物研究所 2021-03-11 WO disclosed