SCHEMBL23099448

SCHEMBL23099448

CN1CCN(c2ccc(C#N)cc2)C=N1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.43
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41
CHRNA10 Q9GZZ6 1/20 0.39
CHRNA9 Q9UGM1 1/20 0.39
KCNH2 Q12809 2/20 0.38
KCNJ1 P48048 1/20 0.38
POLB P06746 1/20 0.37
HRH3 Q9Y5N1 8/20 0.37
NOTUM Q6P988 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP2A6 P11509 1/20 0.35
RAB9A P51151 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24681294 0.77 HRH3 (0.35) HRH3ALDH1A1RAB9A
SCHEMBL21641504 0.74 KDM4E (0.44) CHEK1KDM4ETP53CHRNA10CHRNA9
SCHEMBL23099449 0.73 PRMT6 (0.37) HRH3CYP2A6
SCHEMBL8845493 0.71 LOXL2 (0.36) CHEK1KDM4ETP53CHRNA10CHRNA9
SCHEMBL13876041 0.67 HRH3 (0.42) CHEK1KDM4ETP53CHRNA10CHRNA9
SCHEMBL30639263 0.66 KDM4E (0.47) CHEK1KDM4ETP53CHRNA10CHRNA9
SCHEMBL8845897 0.66 CHRNA10 (0.36) CHEK1KDM4ETP53CHRNA10CHRNA9
SCHEMBL151261 0.66 CHEK1 (0.68) CHEK1KDM4ETP53CHRNA10CHRNA9
Iodide SCHEMBL4213036 0.66 HRH3 (0.41) CHEK1KDM4ETP53CHRNA10CHRNA9
SCHEMBL2384959 0.65 KDM4E (0.80) CHEK1KDM4ETP53CHRNA10CHRNA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021048342-A1 ANTIBACTERIAL COMPOUNDS Janssen Sciences Ireland Unlimited Company (IE) 2021-03-18 WO disclosed