SCHEMBL23102409

SCHEMBL23102409

Cc1c(Br)cccc1-c1nc2c(=O)[nH]ccc2o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
C1R P00736 2/20 0.40
KMT2A Q03164 1/20 0.40
MAPT P10636 3/20 0.38
PARP1 P09874 1/20 0.37
KLK3 P07288 1/20 0.36
TP53 P04637 4/20 0.34
ELANE P08246 1/20 0.34
TOP2A P11388 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
LMNA P02545 2/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
NFKB1 P19838 1/20 0.33
RAB9A P51151 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
USP2 O75604 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23102595 0.78 NPC1 (0.37) KMT2AMAPTTOP2ASMN1; SMN2ALDH1A1
SCHEMBL23102420 0.76 TP53 (0.35) C1RKMT2AMAPTTP53ELANE
SCHEMBL15229119 0.73 PIM1 (0.44) C1RTOP2AF2PLGKLK1
SCHEMBL23102443 0.72 KDM4E (0.43) KMT2AMAPTPARP1ALDH1A1HPGD
SCHEMBL23102399 0.72 PARP1 (0.37) MAPTPARP1TP53ALDH1A1LMNA
SCHEMBL23102583 0.71 USP2 (0.35) KMT2AMAPTTP53TOP2ASMN1; SMN2
SCHEMBL10852717 0.71 MAPT (0.52) C1RKMT2AMAPTTP53ELANE
SCHEMBL23102416 0.69 TP53 (0.31) MAPTTP53TOP2AS1PR1
SCHEMBL15228745 0.69 PIM1 (0.62) KMT2AMAPTTOP2AKDM4ERAB9A
SCHEMBL15228794 0.69 PIM1 (0.58) C1RELANETOP2AF2PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021047555-A1 PREPARATION OF AROMATIC HETEROCYCLIC DERIVATIVE AS IMMUNOMODULATOR AND APPLICATION THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed
WO-2021047556-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME AND USE THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed