SCHEMBL23102420

SCHEMBL23102420

Cc1c(Br)cccc1-c1nc2c(=O)n(C)ccc2o1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.35
SIRT2 Q8IXJ6 3/20 0.35
SIRT1 Q96EB6 3/20 0.35
MAPT P10636 3/20 0.34
C1R P00736 1/20 0.34
KMT2A Q03164 1/20 0.34
ELANE P08246 1/20 0.33
USP2 O75604 2/20 0.33
TOP2A P11388 3/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 2/20 0.33
TSHR P16473 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
NFKB1 P19838 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23102583 0.84 USP2 (0.35) TP53SIRT2SIRT1MAPTKMT2A
SCHEMBL23102416 0.82 TP53 (0.31) TP53MAPTTOP2AS1PR1
SCHEMBL23108686 0.79 TOP2A (0.37) TP53MAPTUSP2TOP2AALDH1A1
SCHEMBL23102479 0.78 PIK3R1 (0.36) TP53MAPTUSP2TOP2AALDH1A1
SCHEMBL23108309 0.78 TNF (0.39) TP53MAPTKMT2AUSP2TOP2A
SCHEMBL23102593 0.77 SMN1; SMN2 (0.41) TP53MAPTUSP2TOP2AALDH1A1
SCHEMBL23102408 0.76 DUT (0.41) USP2
SCHEMBL23102409 0.76 C1R (0.40) TP53SIRT1MAPTC1RKMT2A
SCHEMBL23102594 0.75 TP53 (0.33) TP53MAPTUSP2TOP2AALDH1A1
SCHEMBL23108300 0.75 TNF (0.41) TP53KMT2AUSP2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021047556-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME AND USE THEREOF 上海长森药业有限公司 2021-03-18 WO disclosed