SCHEMBL23116557

SCHEMBL23116557

CN(C)C[C@H](Cc1ccccc1)NC(=O)C(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 4/20 0.48
HDAC6 Q9UBN7 4/20 0.48
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44
ATM Q13315 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MME P08473 3/20 0.44
ACE P12821 1/20 0.44
ACE2 Q9BYF1 1/20 0.44
HDAC1 Q13547 1/20 0.44
RECQL P46063 1/20 0.43
POLB P06746 1/20 0.43
CTRB1 P17538 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21496651 1.00 HDAC4 (0.48) HDAC4HDAC6CYP3A4MAPK1ATM
SCHEMBL21496635 0.84 HDAC4 (0.49) HDAC4HDAC6CYP3A4MAPK1NPC1
SCHEMBL1570133 0.84 HDAC4 (0.49) HDAC4HDAC6CYP3A4MAPK1NPC1
SCHEMBL23116581 0.83 CTRB1 (0.54) HDAC4HDAC6CYP3A4MAPK1NPC1
SCHEMBL23116580 0.83 CTRB1 (0.54) HDAC4HDAC6CYP3A4MAPK1NPC1
SCHEMBL21501009 0.82 ATM (0.67) CYP3A4ATMACE
SCHEMBL21501008 0.82 ATM (0.67) CYP3A4ATMACE
SCHEMBL23116558 0.81 CTRB1 (0.66) HDAC4HDAC6MAPK1ATMNPC1
SCHEMBL10952300 0.81 CTRB1 (0.66) HDAC4HDAC6MAPK1ATMNPC1
SCHEMBL21501067 0.77 CTRB1 (0.68) CYP3A4ATMCTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112312902-B Pd (II) -catalyzed enantioselective C-H arylation of free carboxylic acids 斯克里普斯研究学院 2022-02-18 CN disclosed
US-11021427-B2 Pd(II)-catalyzed enantioselective C—H arylation of free carboxylic acids THE SCRIPPS RESEARCH INSTITUTE (US) 2021-06-01 US disclosed
US-20210087131-A1 PD(II)-CATALYZED ENANTIOSELECTIVE C-H ARYLATION OF FREE CARBOXYLIC ACIDS THE SCRIPPS RESEARCH INSTITUTE 2021-03-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11021427-B2 Pd(II)-catalyzed enantioselective C—H arylation of free carboxylic acids PDCD1, PDK3, PDCD1LG2 HDAC4 1462/4885HDAC6 867/4885CYP3A4 593/4885
US-20210087131-A1 PD(II)-CATALYZED ENANTIOSELECTIVE C-H ARYLATION OF FREE CARBOXYLIC ACIDS PDCD1, PDK3, PDCD1LG2 HDAC4 1480/4885HDAC6 847/4885CYP3A4 594/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.